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1-cyclopentyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(3,5-dimethylphenyl)-4-(4-methyl-1H-pyrrole-2-carbonyl)piperazin-2-one
4-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(azocan-1-yl)-3-(4-{[(3-hydroxypropyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
4-(5-fluoro-2-methylphenyl)-2-methylquinazoline
2-oxo-1-phenyl-N-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-3-carboxamide
4-(oxolan-3-yl)-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole
8-(cyclohex-3-en-1-ylmethyl)-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-oxo-6-(propan-2-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-dihydropyridine-3-carboxamide
1-cyclohexyl-5-{pyrazolo[1,5-a]pyridin-3-yl}-1H-1,2,4-triazole
N4-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N4,6-dimethyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(4-phenylpiperidin-1-yl)acetamide
6,7-dimethoxy-2-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)quinazolin-4-amine
(1S,6R)-9-(2-methyl-1-benzofuran-7-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
2-(4-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}phenoxy)acetic acid
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-({2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
6-chloro-N-[3-(propan-2-yloxy)propyl]-2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}quinazolin-4-amine
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
3-methyl-N-{2-[2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}pyridin-4-amine
7-fluoro-3-({[2-(2-fluorophenyl)ethyl]amino}methyl)-N,N-dimethylquinolin-2-amine
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1,4-oxazepan-6-ol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxy-5-methylbenzamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[4-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethoxy)phenyl]propan-1-one
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(oxolan-2-ylmethyl)benzamide
3-(2-chlorophenyl)-3-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
1-[6-({1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl}oxy)pyridin-3-yl]ethan-1-one
1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-ol
4-(2-ethylphenyl)thiophene-2-carboxamide
3-(2,4-dimethoxybenzoyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
methyl[(1-methylpiperidin-2-yl)methyl][(2,3,4-trimethoxyphenyl)methyl]amine
(1S,5R)-3-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
6-methyl-3-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
5-(3-methoxyphenyl)-4-[1-(3-phenylpropyl)piperidin-4-yl]-2-(pyridin-4-yl)pyrimidine
2-{5-[(2,5-dioxoimidazolidin-4-yl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
6-[(1H-imidazol-2-ylmethyl)(methyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-(3-hydroxypropyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(2S)-2-hydroxypropanoyl]-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
ethyl 4-{[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]amino}piperidine-1-carboxylate
N-[3-(furan-2-yl)propyl]-5-hydroxy-1,2-dimethyl-1H-indole-3-carboxamide
2-{2-[5-(cyclohexylsulfanyl)furan-2-yl]-1H-imidazol-1-yl}ethan-1-ol
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]thiomorpholine
3-{[(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
2-(4-chloro-2-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid