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N-cyclooctyl-1-cyclopentyl-6-oxopiperidine-3-carboxamide
2,3-dimethyl-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-(1-ethylpiperidin-4-yl)-1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethan-1-one
3-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
4-(3,6-dimethylpyrazin-2-yl)-N-(1H-indazol-4-yl)piperazine-1-carboxamide
1-(2-chloro-5-sulfamoylphenyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
(2-methoxyethyl)({2-phenyl-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]ethyl})(pyridin-2-ylmethyl)amine
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-2H-1,3-benzodioxole-5-carboxamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
2-fluoro-6-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
N,2-dimethyl-N-(1,2-oxazol-5-ylmethyl)-1,3-benzothiazole-5-carboxamide
4-({4-methyl-5-[1-(oxan-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-methoxy-1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
4-(hydroxymethyl)-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]azepan-4-ol
N-cyclopropyl-3-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}propanamide
1-[2-(4-benzoylpiperidin-1-yl)-2-oxoethyl]-1,2,3,4,5,6,7,8-octahydroquinolin-2-one
4-(4-ethyl-6-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyrimidin-2-yl)morpholine
N-[3-(4-{[2-(2-chloro-6-fluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-methylfuran-3-carboxamide
4-[3-(benzyloxy)propyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-[2-(butan-2-yloxy)-3-methoxyphenyl]-1H-imidazole
1-(4,7-dimethylquinazolin-2-yl)-N-[2-(2-fluorophenyl)ethyl]piperidine-3-carboxamide
N-(cyclopropylmethyl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-N-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[3-(1-phenylcyclopropyl)-5-[3-(pyridin-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-(1H-indazol-4-yl)-2-(pyrrolidin-3-yl)benzamide
N,N-diethyl-2-{4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
5-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
5-(3,4-dimethylphenoxymethyl)-N-(1-hydroxy-3-methylbutan-2-yl)-1,2-oxazole-3-carboxamide
3-methyl-1-[1-(6-{[(1-methylpiperidin-4-yl)methyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(thiophene-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
(4aS,8aR)-1-propyl-6-(1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[4-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazol-4-yl)thiophen-2-yl]ethan-1-one
1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-[4-(hydroxymethyl)piperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]acetic acid
N-(dicyclopropylmethyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-(morpholin-4-yl)-6-(1H-pyrazol-4-yl)pyrimidin-2-amine
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)quinoxaline-5-carboxamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
4-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)-5,6-dimethylpyrimidine
3-{[1-(2-hydroxyacetyl)pyrrolidin-3-yl]methyl}benzamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(1H-pyrazol-1-yl)acetamide
5-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]pentan-1-ol
N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
N-(3-methylphenyl)-3-{1-[3-(pyridin-2-yl)propanoyl]piperidin-4-yl}propanamide
(3aS,6aS)-2-[(2-aminopyridin-3-yl)methyl]-5-cyclopentanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid