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1-ethyl-2-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-imidazole
N-[2-fluoro-5-(trifluoromethyl)phenyl]-3-oxa-9-azaspiro[5.5]undecane-9-carboxamide
1-(1H-indole-5-carbonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-propoxypropanamide
3-(1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)benzoic acid
N-{3-oxo-3-[3-(4-phenylbenzoyl)piperidin-1-yl]propyl}acetamide
methyl 9-(benzyloxy)-3-{[2-(difluoromethoxy)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
{[4-(difluoromethoxy)phenyl]methyl}[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
8-[(6-methoxynaphthalen-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-{1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-benzyl-3-(diphenylmethyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1,2-oxazole-5-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
2-(2,5-dioxoimidazolidin-1-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
7-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2H-1,3-benzodioxol-5-yl)-5-(5-methoxyfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-methoxy-3-methyl-2-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}-1H-indole
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)-N-propylacetamide
2-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]pyridine-4-carboxamide
2-(3,5-dimethoxyphenyl)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}propanamide
2-[3-(3-methylphenyl)piperidine-1-carbonyl]pyridine
7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-4-(pyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
1-[2-(dimethylamino)-4-{[2-(1H-imidazol-4-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
{[5-(1-cycloheptanecarbonylpiperidin-4-yl)-4-cyclopropyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
4-(2-methoxyethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-[2-(4-methoxyphenyl)ethyl]-4-{[(trimethylpyrazin-2-yl)methyl]amino}pyrrolidin-2-one
(1S,5R)-3-benzoyl-N-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-(2-methoxyethyl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-N3,N3-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
dimethyl(2-{4-[4-(trifluoromethyl)benzoyl]morpholin-2-yl}ethyl)amine
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-ethyl-N-(oxolan-2-ylmethyl)propanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-1-(furan-2-carbonyl)piperidin-3-amine
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-[(4-fluorophenyl)methyl]-N-methylacetamide
N-(2-ethoxyethyl)-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-methoxy-4-[4-(4-methoxybenzoyl)piperazin-1-yl]pyridine-3-carbonitrile
2-[3-(7-methyl-1H-indol-3-yl)phenyl]ethan-1-amine
(3R,4R)-1-[(2E)-2-methylbut-2-en-1-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-[3-(4-{[(1S)-1-carbamoyl-2-phenylethyl]amino}piperidin-1-yl)phenyl]pyridine-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(isoquinoline-3-carbonyl)piperidine-3-carboxylate
4-[4-(6-chloro-1H-1,3-benzodiazol-2-yl)phenyl]-2-methylbut-3-yn-2-ol
5-hydroxy-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]pyrazine-2-carboxamide
4-[({[4-(butan-2-yloxy)-3-ethoxyphenyl]methyl}amino)methyl]-1,2-dihydrophthalazin-1-one
(3-{2-[1-(8-chloroquinolin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1-phenylpyrrolidin-2-one
N-[(3,4-dimethoxyphenyl)methyl]-4-(4-methylphenyl)-N-(pyridin-4-ylmethyl)benzamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide