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4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]-1-[4-(trifluoromethyl)benzenesulfonyl]piperidine
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-phenoxybutan-1-one
4-ethenyl-N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
6-methoxy-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]hexan-1-one
N-[2-(2-fluorophenyl)-1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-6-(methoxymethyl)pyrimidin-4-amine
(2R)-2-amino-3-(furan-2-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
4-[1-(3-phenoxybenzenesulfonyl)azetidin-3-yl]pyridine
6-(1-methyl-1H-pyrazol-4-yl)-1,3-benzothiazol-2-amine
6-(2-hydroxyethyl)-N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-ethyl-1-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl}methyl)urea
N-cyclopentyl-N-propyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(1,5-dimethyl-1H-pyrazol-4-yl)-1-(thiolan-3-yl)urea
8-[3-(4-methoxyphenyl)propanoyl]-1,8-diazaspiro[4.5]decan-2-one
6-ethoxy-2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-1-yl}-4-methylquinazoline
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2-dimethylthieno[3,2-d]pyrimidin-4-amine
N-cyclopropyl-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
{1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-2-(methylsulfanyl)acetamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-2-yl)propanamide
3-{[cyclopropyl(4-methylpyridin-2-yl)methyl]amino}-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
(5S,9aS,9bS)-5-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]-2-cyclopentyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-({2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)pyridine
1-phenoxy-2-[4-(4,4,4-trifluorobutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
3-(2-chlorophenyl)-1-(3-methoxypropyl)-3-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
1-[1-(6-{[2-(dimethylamino)ethyl]amino}pyridine-3-carbonyl)piperidin-3-yl]-3-methylbutan-1-one
4-{3-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(dimethyl-1,2-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
N-[(3S,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
5-methyl-N-[3-(5-methyl-4-{[3-(4-methylphenyl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]thiophene-2-carboxamide
5-(dimethylamino)-2-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
4-[(4-methyl-5-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
5-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidine-1-carbonyl)pyrrolidin-2-one
3-cyclopropyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-oxazole-5-carboxamide
1-ethyl-3-(2-methylpropyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1H-pyrazole-5-carboxamide
2-(2,6-difluorophenyl)-1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
3-[2-(4-fluorophenyl)ethyl]-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
5-(2-aminophenyl)-N-phenylfuran-2-carboxamide
2-(2,3-difluorophenoxymethyl)-N-methyl-N-(3-methylbutyl)-1,3-oxazole-4-carboxamide
N-(1-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
3-methyl-1-(2-methylpropyl)-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-chlorophenyl)-N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
3-methyl-5-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
N-[(3,5-difluorophenyl)methyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-8-carbonyl}cyclopropane-1-carboxamide