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N-[(2-methoxyphenyl)methyl]-N-methyl-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
N-cyclopentyl-2-methyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-1,3-thiazole-4-carboxamide
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
4-{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}benzoic acid
N-[(3R,4S)-1-(2-aminopyrimidin-4-yl)-4-propylpyrrolidin-3-yl]pyrrolidine-1-sulfonamide
2-[(1-ethyl-1H-indol-3-yl)sulfanyl]-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
{3-[(2-fluorophenyl)methyl]-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methanol
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl][(5-cyclopropyl-1,2-oxazol-3-yl)methyl]methylamine
2-benzyl-8-(2,3-difluorobenzoyl)-2,8-diazaspiro[4.5]decan-3-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
(4aR,8aS)-1-[3-(dimethylamino)propyl]-6-(3-methoxybenzoyl)-decahydro-1,6-naphthyridin-2-one
2-methyl-6-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
3-methoxy-2-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
7-[(2-fluorophenyl)methyl]-2-[(2-methoxypyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-({1-[(3-methylphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}methyl)morpholine
2,5-dimethyl-3-(4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazin-1-yl)pyrazine
methyl 4-[5-(3-phenoxypropanamido)-1H-pyrazol-1-yl]piperidine-1-carboxylate
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
2-(2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)-N-methylacetamide
N3-[(2,6-difluoro-3-methylphenyl)methyl]-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(3-chlorophenyl)-4-cyclobutanecarbonylpiperazin-2-one
2-{[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}-4-methoxyphenol
2-(3-methoxyphenyl)-1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethoxy]ethan-1-ol
6-tert-butyl-2-(3-{[(2-hydroxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(thiophene-2-carbonyl)piperazine
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(2-methylphenyl)methyl]piperazine
(2S,4S)-N-ethyl-1-[(2-fluorophenyl)methyl]-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
2-methyl-6-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,3-benzothiazole
1-cyclopropyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-6-oxopiperidine-3-carboxamide
1-(2-methoxyethyl)-8-[(4-methylphenyl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-2,3-dihydro-1H-isoindole-2-carboxamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylic acid
(1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-yl)methanol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-[3-(furan-2-yl)phenyl]-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine-4-carboxamide
3-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-2H-chromen-2-one
2-[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
3-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
N-cyclohexyl-N-(thiophen-3-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
N-ethyl-N-methyl-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]acetamide
N-cyclohexyl-N-(pyridin-2-ylmethyl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
(2S,4S)-4-amino-1-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-(oxan-4-yl)benzamide
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-4-carboxamide