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1-(6-methoxypyrimidin-4-yl)-4-[3-(morpholin-4-yl)propyl]-1,4-diazepane
4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-[(6-ethoxypyridin-3-yl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[(5-methylpyrazin-2-yl)methyl]-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-(4-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}phenyl)acetamide
methyl 6-(2-methylbutanoyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[1-(2,3-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]butanoic acid
3-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-N,N-dimethylaniline
(3S,9aR)-8-(4-chlorobenzenesulfonyl)-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
9-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
methyl (2S,4R)-4-(3-hydroxynaphthalene-2-amido)-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxylate
3-(4-fluorophenoxymethyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N,N-diethylpropanamide
dimethyl(2-{2-[1-(pyridine-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-(3-{4-[(2-acetamido-3-methylbutanamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-2,5-dimethylfuran-3-carboxamide
2-(3-fluoro-5-methylphenyl)-N-(propan-2-yl)pyridine-4-carboxamide
4-{[3-(methylsulfanyl)phenyl]methyl}-1,4-oxazepan-6-ol
1-{2-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]ethyl}-6-methyl-1,2-dihydropyridin-2-one
ethyl 4-{[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}piperidine-1-carboxylate
2-methoxyethyl 7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxylate
4-[({4-methyl-5-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]pyridine
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
5-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{4-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]piperazin-1-yl}-N-ethylacetamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[(3-methoxyphenyl)methyl]amine
N-(piperidin-4-yl)-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(butan-2-yl)-3-acetamido-N-(pyridin-3-ylmethyl)benzamide
1-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
2-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)benzoic acid
3-[1-(4-chloro-2-hydroxybenzoyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]propanamide
(1S,5R)-3-(1,3-benzothiazole-6-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
benzyl(cyclobutylmethyl){[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}amine
2-{[6-(cyclohex-1-en-1-yl)quinazolin-4-yl]amino}ethan-1-ol
N-(2,3-dihydro-1H-inden-2-yl)-5-(1H-indol-1-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-(2-methoxyethyl)-4-(piperidin-3-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[3-(propan-2-yloxy)propyl]benzamide
2-(2-fluorophenoxymethyl)-N-[(2R)-1-hydroxybutan-2-yl]-1,3-oxazole-4-carboxamide
methyl 3-cyclobutaneamido-5-{[(4-fluoro-3-methoxyphenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-ethyl-1-methyl-5-(morpholine-4-carbonyl)-1H-1,3-benzodiazol-7-yl]-2-methoxybenzamide
methyl 3-[({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)carbamoyl]propanoate
2-[1-(2-phenylethyl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
4-({1,9-dioxaspiro[5.5]undecan-4-yl}sulfamoyl)-N-methylthiophene-2-carboxamide
(2S)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]pyrrolidine-2-carboxamide
2-(3-fluorophenoxymethyl)-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-oxazole
ethyl 4-[6-(5-methylthiophene-2-carbonyl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-4-[2-(methylsulfanyl)pyrimidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]amine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-methylfuran-2-carboxamide
3-({[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]oxy}methyl)pyridine