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3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-1-(4-methylpiperidin-1-yl)propan-1-one
1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-N-cyclopropylpiperazine-2-carboxamide
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
N-[1-(1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)piperidin-4-yl]methanesulfonamide
N-[(4-chlorophenyl)methyl]-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
2-benzyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1,3-thiazole-4-carboxamide
N-[(2-fluorophenyl)methyl]-3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanamide
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
3-chloro-5-[2-(3-methoxypropyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
7-methanesulfonyl-4-methyl-2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]quinazoline
(3S,4S)-4-(pyrrolidin-1-yl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-ol
2-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]piperidine
1-(2,2-dimethylpropyl)-4-{[(4-fluoro-3-methoxyphenyl)methyl]amino}pyrrolidin-2-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-2-carboxamide
8-[(2-chlorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-7-fluoro-N-(2-hydroxyethyl)-3-methyl-1-benzofuran-2-carboxamide
3-ethyl-1-{2-[4-(pyridin-2-ylmethyl)morpholin-2-yl]ethyl}urea
N-(oxan-4-yl)-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(1S,5R)-3-(pyridin-2-ylmethyl)-6-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
3-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluorobenzamide
1-benzoyl-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1,3-oxazole-4-carboxamide
N-[1-benzyl-2-methyl-7-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
3,7-dimethyl-11-(2,4,5-trimethoxybenzoyl)-3,7,11-triazaspiro[5.6]dodecane
8-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl]{[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
2-cyclopentyl-N-[(3R,4S)-4-cyclopropyl-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]acetamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
8-[(2,4-difluorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,6R)-9-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N4-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-5,6-dimethylpyrimidine-2,4-diamine
4-[1-(7-fluoro-4,6-dimethylquinazolin-2-yl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
6-(4-aminopiperidin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-4-yl)-3-methyl-4H,5H,6H,7H-[1,2]oxazolo[5,4-b]pyridin-6-one
ethyl 4-{6-[(2,4-dimethoxy-3-methylphenyl)methyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-(1,2-oxazinan-2-yl)propanamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
3-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1,9-dimethyl-4-(6-methyl-2-phenylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]propan-1-one
3-[2-({[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]carbamoyl}amino)phenyl]-N-methylpropanamide
{4-[4-(pyridin-3-yl)pyrimidin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(pyrimidin-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(5-methylfuran-2-yl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[1-(3-methoxypropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]methyl}-N,N-dimethyl-1,2,4-oxadiazole-5-carboxamide