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3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
N-(4-fluorophenyl)-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-3-amine
N-cyclopropyl-1-[(1s,4s)-4-(4-methylbenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-methoxypyrazine
N-[4-(8-hydroxyquinolin-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]methanesulfonamide
1-cyclopropyl-1-[(3-hydroxyphenyl)methyl]-3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
1-(2-methoxyethyl)-5-[2-(naphthalen-1-yl)acetyl]-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-2-yl)piperazine
1-(3-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}propyl)piperidine-4-carboxamide
1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-4-benzylpiperidin-4-ol
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-(4-aminopyrimidin-2-yl)-3-(2-phenylethyl)piperidine-3-carboxylic acid
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(3-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
3-{2,7-diazaspiro[4.5]decan-7-yl}-N-(2,4-dimethylphenyl)-3-oxopropanamide
2-fluoro-N-({8-[3-(methylsulfanyl)propanoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
(1S,5R)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-[1-(thiophen-2-yl)ethyl]acetamide
4-cyclopentyl-6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[(2S,4R)-1-[(2,6-difluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
2-[(4-methoxyphenyl)methyl]-1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
4-[(2-methoxyphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-ethoxy-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1,3-oxazole-5-carboxamide
3-(4H-1,2,4-triazol-4-yl)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-(2-methoxyethyl)pyrrolidine
[(4,6-dimethylpyridin-2-yl)methyl][(5-ethylpyridin-2-yl)methyl]methylamine
1-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)pyrrolidin-2-one
methyl 5-{2-methylthieno[2,3-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
ethyl 3-[(2-fluorophenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylate
7-[(6-chloro-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[3-(diphenylmethyl)-1,2-oxazole-5-carbonyl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-(2,6-dimethoxypyridin-3-yl)acetic acid
[1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
3-chloro-N-(2-methoxyethyl)-4-({1-[4-(methylsulfanyl)butan-2-yl]piperidin-4-yl}oxy)benzamide
(3R,4S)-3,4-dimethyl-1-(5-phenyl-1,2-oxazole-4-carbonyl)piperidin-4-ol
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-({4-[3-(dimethylamino)propoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[(2-chlorophenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{2-[(4aS,8aR)-decahydroisoquinolin-2-yl]-2-oxoethyl}-5-(dimethylamino)-2,3-dihydropyridazin-3-one
ethyl 1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-imidazole-2-carboxylate
2-methyl-6-[3-(propan-2-yl)-5-(1,2,3-thiadiazol-4-yl)-1H-1,2,4-triazol-1-yl]-1,3-benzothiazole
N-methyl-N-{2-phenyl-1-[1-(quinolin-7-ylmethyl)piperidin-4-yl]ethyl}thiophene-2-carboxamide
1-(4-chlorophenyl)-4-[2-(4-methoxyphenyl)acetyl]-5-methylpiperazin-2-one
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
methyl 1-(2-methoxyethoxy)-8-[(2-methoxyphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-methyl-4-{4-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}butan-2-ol
N-({7-[2-(3,4-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide