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1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
3-{[1-(1-butanoylpiperidin-4-yl)pyrrolidin-3-yl]methyl}benzoic acid
4-[(3-methylphenyl)sulfanyl]-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
6-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
ethyl 2-[1-(thiophene-3-sulfonyl)piperidin-2-yl]acetate
2-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-6-fluoroquinoline
3-[(1R,2S)-2-hydroxycyclohexyl]-3-methyl-1-[3-(2-methylphenyl)phenyl]urea
(4aS,7aR)-1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-hydroxy-4-methoxybenzamide
(2S)-2-({2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-inden-2-yl}formamido)-4-methylpentanamide
1-[4-(8-methyl-2-{[methyl({[2-(trifluoromethyl)phenyl]methyl})amino]methyl}quinazolin-4-yl)piperazin-1-yl]ethan-1-one
5-methyl-1-(1,2-oxazol-5-ylmethyl)-5-phenylpiperidin-2-one
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-benzyl-3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-{5-[1-(furan-3-ylmethyl)-1H-1,2,3-triazol-4-yl]furan-2-yl}benzonitrile
6-fluoro-N-(1-hydroxybutan-2-yl)-2-oxo-N-(thiophen-2-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
2-[1-methyl-10-oxo-4-(thiophen-2-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-3-ylmethyl)amino]ethyl]piperidin-1-yl}ethan-1-one
2-(2,5-dimethylfuran-3-carbonyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
N-(2-benzylbutyl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
8-[(3-chlorophenyl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-{[(2-methoxy-2-methylpropyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2-(1-ethylpiperidin-4-yl)-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
(2-{2-[1-(2,5-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
3-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-[(2-propyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-(2H-indazol-2-yl)-1-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
4,6-dimethyl-3-[2-(3-phenylpropyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
2-[N-methyl-1-(3,4,7-trimethyl-1H-indol-2-yl)formamido]-2-(pyridin-3-yl)acetic acid
2-chloro-5-({[1-(1-methyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-methanesulfonyl-decahydro-1,6-naphthyridin-2-one
N'-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N'-methylbutanediamide
7-methyl-N-[3-(methylsulfanyl)phenyl]-3,7,11-triazaspiro[5.6]dodecane-11-carboxamide
5-(4-cyclohexylpiperazine-1-carbonyl)-4-methyl-2-(pyridin-3-yl)pyrimidine
(3R,9aR)-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[(2-methyl-1H-imidazol-1-yl)methyl]-1-[4-(methylsulfanyl)phenyl]-1H-1,2,4-triazole
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-[(4-methylphenyl)sulfanyl]piperidine
3-(2H-1,3-benzodioxol-5-yl)-1-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
N-(2,2-dimethyloxan-4-yl)-3-(diphenylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
9-methoxy-10-(pyrrolidine-1-carbonyl)-3-(quinolin-5-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-(2-chloro-4-{[methyl(thian-4-yl)amino]methyl}phenoxy)propanoic acid
2-cyclohexyl-N-{7-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}acetamide
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
8-[(3-hydroxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(dimethylamino)methyl]-N-{2-[2-(propan-2-yloxy)phenyl]ethyl}benzamide