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(4R,6S)-4-methyl-6-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}-1,3-diazinane-2-thione
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methyl-N-(2-phenylethyl)propanamide
1-[(3-fluorophenyl)methyl]-4-(2-methylpyridin-4-yl)piperazine
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-7-methylquinoline
4-ethyl-6-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(pyrrolidin-1-yl)pyrimidine
N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-propyl-1H-pyrazole
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
(2R,3R,6R)-3-(4-fluorophenyl)-5-(3-propyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2,3-dihydro-1H-inden-2-yl)-4-{[(2-methoxyphenyl)methyl]amino}pyrrolidin-2-one
(1R,2R,6S,7S)-4-[2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
benzyl 3-({[1-(propan-2-yl)-1H-pyrazol-4-yl]carbamoyl}amino)pyrrolidine-1-carboxylate
(1S,5R)-3-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]acetamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-(naphthalen-1-ylmethyl)acetamide
3-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-1-(3-methoxyphenyl)urea
1-[5-(5-chlorofuran-2-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
1-(1-cyclooctylpiperidin-3-yl)-4-phenylpiperazine
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
6-(4-fluorophenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7-(3-methylbut-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
9-[(2S)-2-amino-2-cyclopropylacetyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-ethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrimidin-2-amine
N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]-2-(piperidin-4-yl)acetamide
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-5-propyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
methyl (2S,3S)-2-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}formamido)-3-methylpentanoate
methyl 8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methyl-1H-1,3-benzodiazole-4-carboxamide
N-(2-phenylethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-ethyl-4-{2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperazin-2-one
6-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methoxy-N,N-dimethyl-5-({[3-(2-oxopyrrolidin-1-yl)propyl]carbamoyl}amino)benzamide
{[4-(2-{4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)(quinolin-6-ylmethyl)amine
3-(1H-1,3-benzodiazol-1-yl)-1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]propan-1-one
1-{5-[(4-benzylpiperazin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}azocane
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(2-oxopyrrolidin-1-yl)benzamide
1-[2-(piperazin-1-yl)ethyl]-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-1,2,3-triazole-4-carboxamide
3-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
1-methanesulfonyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-amine
[3-(1H-imidazol-4-ylmethyl)-9-[(2-methoxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-(4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
9-[2-(4-fluorophenoxy)ethyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2R,3R)-1'-[(2,3-difluorophenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-{5-[(cycloheptylamino)methyl]-2-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
3-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidine-1-carbonyl)pyridine
N-{3-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]phenyl}propanamide
1-methyl-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine