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(1S,5R)-1,3,3-trimethyl-6-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-6-azabicyclo[3.2.1]octane
(2S)-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
5-methoxy-9-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(4-methylpiperazin-1-yl)propyl]acetamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-indazole-3-carboxamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[4-(2-methylpropyl)benzoyl]-1,4-diazepan-5-one
2-methyl-5-(4-{[4-(1,2,3-thiadiazol-4-yl)phenyl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-(oxan-4-ylmethyl)-4-[2-(phenylsulfanyl)acetyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[1-(3-fluorobenzoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
4-hydroxy-N-pentyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
methyl 6-{[bis(prop-2-en-1-yl)amino]methyl}-3-[2-(2-fluorophenyl)acetamido]thieno[2,3-b]pyridine-2-carboxylate
(1S,5R)-6-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(2-methoxyphenyl)methyl]-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2,5,6-trimethylpyrimidine
1-(2-methoxyethyl)-4-(4-phenyl-1H-imidazol-5-yl)piperidine
2-amino-3-ethyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[(2-fluorophenyl)methoxy]-8-[(2E)-2-methylbut-2-en-1-yl]-1,8-diazaspiro[4.5]decan-2-one
methyl (2S)-1-(2-{1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl}acetyl)pyrrolidine-2-carboxylate
1-[(2-methylphenyl)methyl]-4-(piperidin-3-ylmethyl)piperazine
3-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]phenol
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
(2-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-1,3-thiazol-4-yl)methanol
(1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
methyl 2-[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]pyridine-3-carboxylate
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-(propan-2-yl)acetamide
(3S,4S)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-3-ol
3-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-ethoxy-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-cyclopentyl-2-methyl-N-(3-phenylprop-2-yn-1-yl)imidazo[1,2-a]pyrimidine-3-carboxamide
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-tert-butyl-1-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
1-(3-methanesulfonamido-4-methoxyphenyl)-3-methyl-3-[1-(1,3-thiazol-2-yl)ethyl]urea
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-2,3,4-trimethoxy-N-(pyridin-3-ylmethyl)benzamide
7-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoacetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
7-[(4-fluorophenyl)methyl]-2-(3-propyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
1-(2-phenoxypropanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(4-methoxyphenyl)pyridine-3-carbonitrile
4-methyl-1-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentane-1,2-dione
1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)-2-phenoxyethan-1-one
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-hydroxyethyl)-N-methylacetamide
4-fluoro-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
(3R,5S)-N3-(4-fluorophenyl)-1-(2-methylpropyl)-N5-(2-phenoxyethyl)piperidine-3,5-dicarboxamide
2-(furan-2-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}azepane
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(pyrrolidin-1-yl)benzamide
1-[2-(dimethylamino)ethyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
5-(6-methoxy-3-methyl-1-benzofuran-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
methyl (2S,3S)-2-({1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazol-7-yl}formamido)-3-methylpentanoate
(3S,4S)-1-(pyridin-4-ylmethyl)-4-(thiomorpholin-4-yl)pyrrolidin-3-ol
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine