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2-[3-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-methoxypyrimidine
3-{2-[6-methoxy-3-oxo-4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
6-methyl-4-[3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-(cyclopropylmethyl)-5-(3,4-dimethoxybenzoyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S)-2-amino-1-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-4-(methylsulfanyl)butan-1-one
5-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(1R,5R)-6-[(2-cyanophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}formamido)-4-(methylsulfanyl)butanoic acid
4-{1-[2-(oxolan-3-yl)ethyl]-1H-imidazol-2-yl}quinoline
N-[(3R,4S)-4-cyclopropyl-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
methyl 3-[(2,6-difluorophenyl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-5-(4-methoxyphenyl)-N-(pyridin-4-ylmethyl)furan-2-carboxamide
N-(dicyclopropylmethyl)-N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-[2-(cyclohex-1-en-1-yl)ethyl]-4-[4-(1H-imidazol-1-yl)phenyl]-1H-1,2,3-triazole
2,6-difluoro-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-methylbenzamide
1-(4-aminopyrimidin-2-yl)-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
N-benzyl-N-methyl-1-(6-methylpyridine-2-carbonyl)piperidin-3-amine
(1R,5R)-6-(7-fluoro-2-methylquinoline-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(4-methoxy-2-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-chlorobenzenesulfonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-2,3-dimethoxy-N-(oxolan-2-ylmethyl)benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(2-oxopiperidin-1-yl)butanamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(methylcarbamoyl)methyl]propanamide
1-ethyl-5-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-N-phenylpiperidine-1-carboxamide
N3-cycloheptyl-1-cyclopropyl-N5-[2-(3-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
2-fluoro-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)benzamide
1-{4-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
[(3R,4S)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(3aR,6aR)-2-cyclopentyl-5-[(1-ethyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2R,3R)-2-ethoxy-1'-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-(2-hydroxyethyl)piperidine-3-carboxamide
2-{3-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]propyl}-2,3-dihydro-1H-isoindole-1,3-dione
(4aR,8aS)-6-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
7-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(2-methylpropyl)-3-propanamido-N-(pyridin-2-ylmethyl)benzamide
3-methyl-5-{5-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1,2-oxazole
1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-(piperidine-1-carbonyl)piperidine
1-{[1-(2-hydroxyethyl)piperidin-3-yl]methyl}-3-[2-(3-methoxyphenyl)phenyl]urea
4-{1-methyl-4-[4-(piperidin-1-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
3-hexyl-8-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-({1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octan-6-yl}methyl)-2,6-dimethoxyphenol
2-(3-chlorophenoxy)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)({[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl})methylamine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
2-(dimethylamino)-N-[(4-methoxyphenyl)methyl]-4-methyl-N-propylpyrimidine-5-carboxamide
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(pyrrolidin-1-yl)propyl]amine
1-methyl-4-[(5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)methyl]piperidine