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5-(5-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}furan-2-yl)-1H-pyrazole
N-methyl-5-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2,2-dimethyl-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
7-(2-hydroxyethyl)-2-(1-phenylpiperidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{1-[(tert-butylcarbamoyl)methyl]piperidin-3-yl}benzoic acid
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(morpholin-4-yl)ethyl]acetamide
6-(4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)quinoxaline
7-(piperidine-1-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(furan-2-ylmethyl)-N-(isoquinolin-5-ylmethyl)-N-methylpiperidine-3-carboxamide
1-{2-[2-(5-propylfuran-2-yl)-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
6-methyl-N4-[3-(4-methylpiperazin-1-yl)butyl]pyrimidine-2,4-diamine
8-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-(3,4-dimethylphenyl)-6-fluorobenzamide
N-methyl-1-oxo-N-[1-(pyridin-3-yl)propyl]-1,2-dihydroisoquinoline-4-carboxamide
ethyl 4-{6-[(3,5-dimethoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
(3aR,6aS)-N-{3-[2-(dimethylamino)acetamido]-4-methylphenyl}-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
5-[1-tert-butyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-2-methylpyrimidine
2-{1-cyclohexyl-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{2-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)carbamoyl)amino]phenyl}-N,N-dimethylacetamide
(1-benzothiophen-2-ylmethyl)({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)amine
5-chloro-N-[2-(dimethylamino)ethyl]-N-ethyl-3-phenyl-1H-indole-2-carboxamide
6-chloro-3-({[(2,2-dimethyl-1-phenylcyclopropyl)methyl]amino}methyl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
5-(4-fluorophenyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
[(3R,5R)-1-(3-chloro-4-methylbenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
6-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}pyridine-3-carboxylic acid
methyl 4-{[1-(3-phenylpropyl)piperidin-3-yl]carbamoyl}benzoate
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
2-(1-methyl-1H-imidazol-2-yl)-1-(2,2,6-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1H-imidazole
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(3,4-dimethoxyphenyl)propanamide
4-(2-fluoro-4-methylbenzoyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-chloro-2-({[cyclopropyl(pyridin-2-yl)methyl](methyl)amino}methyl)quinolin-4-ol
4-methyl-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}pentanamide
(2S,4R)-N-methyl-1-(thiophen-3-ylmethyl)-4-[3-(1H-1,2,4-triazol-1-yl)propanamido]pyrrolidine-2-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-4-methyl-1,3-oxazole-5-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
8-(9H-purin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(adamantan-1-yl)-N-cyclopropyl-4-hydroxy-N-(2-methylpropyl)pyrimidine-5-carboxamide
3-butyl-1-methyl-4-(2,6,8-trimethylquinoline-4-carbonyl)piperazin-2-one
3-ethyl-3-(hydroxymethyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
3-(3-methylbutyl)-8-[1-(1H-pyrazol-1-yl)propan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aS,8aS)-2-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-decahydroisoquinolin-4a-ol
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)pyrimidin-2-amine
3-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-(2-chlorobenzenesulfonamido)-5-{[2-(thiophen-2-yl)acetamido]methyl}benzoate
3-(4-{3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}piperazin-1-yl)propanamide
N-{2-[3-(propan-2-yloxy)phenyl]ethyl}oxolane-3-carboxamide