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2-[5-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-ethyl-6-(3-fluorophenyl)-N-(oxolan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3S,4R)-4-(2-methylphenyl)-1-(trimethyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
4-{3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2-{bis[(3-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
1-(dimethylamino)-2-(4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
1-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
3-(2,5-dioxoimidazolidin-4-yl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]propanamide
(1R,5R)-6-(3-phenoxypropyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{3-[3-(4,6-dimethoxypyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
2-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(2H-1,3-benzodioxol-5-ylformamido)methyl]-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
(1R,5S,8S)-8-methoxy-3-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-3-azabicyclo[3.2.1]octane
7-(quinolin-2-ylmethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
5-(furan-2-yl)-3-[(4-phenyl-5-propyl-1H-imidazol-1-yl)methyl]-1,2-oxazole
ethyl 1-[(4-methoxyphenyl)methyl]-5-[2-(pyridin-4-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,5,7-trimethyl-3,7-diazabicyclo[3.3.1]nonane
2-(3-methylphenyl)-N-(1-{3-[4-(pyrazin-2-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
(3aR,6aS)-5-[(5-cyclohexylthiophen-2-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(furan-3-ylmethyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
2-amino-6-(4-hydroxyphenyl)-4-[2-(methoxymethyl)pyrimidin-5-yl]-5-methylpyridine-3-carbonitrile
4-(dimethylamino)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-[5-(3-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1λ6-thiane-1,1-dione
N-{[1-(3-cyclopentylpropyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
1-(2-chloro-4,6-dimethylphenyl)-3-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]urea
8-(3-methylbutyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-chloro-2-fluoro-N-[2-(6-methylpyridin-2-yl)ethyl]benzamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(4-chlorophenyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
methyl (2S,4S)-1-[(2-chlorophenyl)methyl]-4-(furan-2-amido)pyrrolidine-2-carboxylate
1-(2-ethoxyethyl)-N-(oxan-4-yl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-[1-(2,2-diphenylacetyl)piperidin-4-yl]-5-methyl-3-(pyridin-4-ylmethyl)imidazolidine-2,4-dione
N-[(8-{[3-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]benzamide
N-methyl-3-[4-(3-methylphenyl)piperazin-1-yl]-N-(thiophen-3-ylmethyl)propanamide
2-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-3-methylpyridine
3-phenyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
1-(3-methoxyphenyl)-4-(5-methyl-1H-indazole-3-carbonyl)piperazin-2-one
methyl 1-ethoxy-8-[(4-methoxy-2,5-dimethylphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-methoxy-5-{[4-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
4-{1-[(6-methoxynaphthalen-2-yl)methyl]azetidin-3-yl}morpholine
4-{4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-N-(1-phenylethyl)benzamide
1-(2-methoxyphenyl)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperazin-2-one
8-({1-[(4-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[7-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}benzenesulfonamide
4-(4-ethoxyphenyl)-2-(4-methanesulfonylphenyl)-1H-imidazole
1-methyl-2-oxo-8-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{2-oxo-2-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione