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2-(furan-2-yl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
N5-[1-(2-chlorophenyl)ethyl]-1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
5-[(4-chlorophenyl)methyl]-5-{3-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2-methyl-8-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-(6-methoxypyridin-3-yl)-4-methylbenzamide
methyl 3-acetamido-5-{[(3-methylthiophen-2-yl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(1H-indol-3-yl)-1-[3-(methoxymethyl)pyrrolidin-1-yl]butan-1-one
1-methyl-4-{5-[(3-propoxypiperidin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1,4-diazepane
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-N-phenylpyrimidin-2-amine
2-{1-[(2-methylphenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[(2,3-dimethoxyphenyl)methyl]-3-(4-methylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-(1-{[4-(furan-2-yl)phenyl]methyl}pyrrolidin-2-yl)-5-methyl-1,2-oxazole
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
4-(5-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
1-[benzyl(methyl)amino]-3-(4-{[(cyclopropylmethyl)amino]methyl}phenoxy)propan-2-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
2-(carbamoylamino)-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
N-(3-acetylphenyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
3,3-dimethyl-1-{[5-(piperidin-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
N-{[5-fluoro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenoxypropanamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N-[1-(methoxymethyl)cyclopentyl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-[3,5-dimethyl-1-(2-oxopropyl)-1H-pyrazol-4-yl]benzoic acid
(3aS,7aR)-2-(3-chloro-4-methylbenzoyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-[3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]pyridine
5-(3,5-dichloro-4-methylbenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(1,2-benzoxazol-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
1-cyclohexyl-N3-[2-(4-fluorophenyl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
{1-[(3-chloro-4-ethoxyphenyl)methyl]-3-propylpiperidin-3-yl}methanol
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methylpyrazine-2-carboxamide
(3R,4S)-1-(2,5-dimethylpyrimidin-4-yl)-4-propylpyrrolidin-3-amine
1-[2-(cyclohex-1-en-1-yl)ethyl]-4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
3-({3-[hydroxy(phenyl)methyl]-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-1,3-oxazolidin-2-one
N-(2,4-dimethylphenyl)-2-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)acetamide
N-[(3-{2-[(dimethylamino)methyl]phenyl}phenyl)methyl]acetamide
4-amino-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}pyridine-2-carboxamide
4-{4-phenyl-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazol-5-yl}phenol
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-imidazole-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)(quinolin-8-ylmethyl)amine
2-methyl-4-{5-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}but-3-yn-2-ol
2-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-ethyl-N-(1H-indol-2-ylmethyl)-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-(2,6-dimethylpyridin-3-yl)-N-[1-(4-methylpyridin-2-yl)propyl]pyrimidin-2-amine
5-(2-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione