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3-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methylpropanamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(3-fluorophenyl)propanamide
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
1-ethyl-N,3-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(1H-imidazol-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
(4aS,8aR)-1-(3-aminopropyl)-6-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
3,5-dimethyl-N-{3-methyl-1-[7-(quinolin-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
1-(4-{[2-(4-fluorophenyl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(3R,5S)-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-phenylacetamide
5-(methoxymethyl)-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,3,4-oxadiazole-2-carboxamide
1-[(4-fluorophenyl)methyl]-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-(propan-2-yl)-1,4-diazepane
7-(2H-1,3-benzodioxole-5-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(3,5-dimethylbenzoyl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-(4-chlorophenyl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropane-1-carboxamide
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-indazole-3-carboxamide
N-methyl-2-(morpholin-4-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrimidine-5-carboxamide
(2R,3S,6R)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 1-[1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carbonyl]piperidine-2-carboxylate
4-ethyl-5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-3-carboxylic acid
(3S,4S)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(3-phenylpropyl)-N-[2-(pyridin-3-yloxy)propyl]-1,3-benzoxazole-5-carboxamide
3-ethyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-(morpholin-3-yl)acetamide
N-benzyl-6-[4-(piperidin-1-ylmethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(furan-2-ylmethyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]piperidine-4-carboxamide
N-{[7-(1-phenylcyclopropanecarbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
6-methyl-2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pyridine-3-carbonitrile
4-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-1-(cyclopropylmethyl)-2-(propan-2-yl)-1,4-diazepane
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(3-methoxypropyl)benzamide
4-{2-[2-(methylamino)ethoxy]phenyl}-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{[3-(1H-imidazol-1-yl)propyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
5,7-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-(2-methylprop-2-en-1-yl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
3-(4-methyl-1H-pyrazol-5-yl)-1-[(2,3,6-trifluorophenyl)methyl]piperidine
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(diethylamino)propanamide
2-(butylsulfanyl)-N4-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrimidine-4,6-diamine
2-(pyridin-2-yl)-5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
5-phenyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,2,4-triazin-3-amine
(1R,2S,4R)-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
[2-(1H-imidazol-1-yl)ethyl](methyl){[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
N-[(2-fluorophenyl)methyl]-2-(3-hydroxyadamantan-1-yl)-N-(2-methoxyethyl)acetamide
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-(4-fluorophenyl)-N-(2-{7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
2-(methoxymethyl)-6-methyl-1-(naphthalen-1-ylmethyl)-3-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}-1,4-dihydropyridin-4-one