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3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]propanamide
1-(2,3-dihydro-1H-inden-5-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-amine
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1,2-oxazole-3-carboxamide
(5-{[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
3-fluoro-5-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-ethyl-3-(pyridin-2-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-[(4-methylphenyl)sulfamoyl]-6-(pent-4-enoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 3-[(2-methylphenyl)methyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(6-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrimidin-4-yl)piperidin-4-ol
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylcyclopropane-1-carboxamide
1-(2,1-benzoxazole-3-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-{1-[(2E)-3-(4-chlorophenyl)prop-2-enoyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
N,N-diethyl-1-{5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperidine-3-carboxamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-{imidazo[1,2-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
5-(2,1,3-benzothiadiazol-5-ylmethyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5,6-dimethyl-3-{4-[2-(4-methylphenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
methyl 5-(3-{[(3,5-dimethoxyphenyl)formamido]methyl}piperidin-1-yl)-5-oxopentanoate
2-phenyl-1-[1-(quinolin-4-ylmethyl)piperidin-3-yl]ethan-1-one
(2R,6R)-4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
1-(2-amino-9H-purin-6-yl)-4-butyl-1,4-diazepan-6-ol
7-(2-methoxyacetamido)-N,1-dimethyl-2-phenyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
N-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
3-(2-methylpropyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-oxazole-5-carboxamide
{3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-oxopropyl}urea
2-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-5-(dimethylamino)-2,3-dihydropyridazin-3-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
(3S,4R)-1-(2,6-dimethoxypyridine-3-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
(3R,5S)-5-{4-[2-(pyridin-4-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-3-amine
5-[2-(4-fluorophenyl)azetidine-1-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
2-(2-methoxyethyl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-benzoxazole-6-carboxamide
1,3-dimethyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-3-carboxamide
N-(2-fluoroethyl)-3-{[2-oxo-2-(piperazin-1-yl)ethyl]sulfamoyl}benzamide
N-(pyridin-2-ylmethyl)-3-{[1-(pyrimidin-2-yl)piperidin-4-yl]oxy}benzamide
2-[(3-methoxyphenyl)amino]-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}butanamide
1-[3-(1,4-diazepane-1-sulfonyl)benzoyl]piperidine-4-carbonitrile
6-methyl-1-{3-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(quinolin-6-ylmethyl)acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
1-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
N-(furan-2-ylmethyl)-6-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
2-acetyl-8-[(1-ethyl-1H-indol-6-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(piperidin-3-yl)benzamide
1-[(6-methoxypyridin-3-yl)methyl]-3-phenylpyrrolidin-3-ol
7-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-{[4-(5-carbamoylpyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid