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N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)oxolane-2-carboxamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[3-(4-methyl-1,3-thiazol-5-yl)propyl]amine
4-ethyl-1-methyl-3-{1-[(8-methylquinolin-5-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}piperazin-2-one
N-[3-(methylsulfanyl)propyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-2-[methyl({[(2R,5S)-5-{[6-(trifluoromethyl)pyridin-3-yl]methyl}oxolan-2-yl]methyl})amino]acetamide
3-[(1-{imidazo[1,2-a]pyridine-3-carbonyl}pyrrolidin-3-yl)methyl]benzamide
(2R,6R)-4-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-methyl-N-(2-phenylethyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{1-[2-(diethylamino)ethyl]-1H-1,2,3-triazol-4-yl}phenol
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
3-(2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
2-methyl-9-[3-(2-methylphenyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-cyano-2-fluorophenyl)-3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}urea
1-{6-hydroxy-4-[5-(methoxymethyl)thiophene-2-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
2-{4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyrimidin-2-yl}phenol
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
5-methyl-1'-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,7aR)-1-[(3,5-dimethylphenyl)methyl]-4-(1H-imidazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[9-(cyclopropylmethyl)-3-(5-methyl-1,3-oxazole-4-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
6-(2,3-dihydro-1-benzofuran-7-yl)-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
N-methyl-2-(4-propanoylphenoxy)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
(2R,3R,6R)-5-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-(2-methoxyethyl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(thiophen-2-ylmethyl)acetamide
(3R,4S)-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-3,4-dimethylpiperidin-4-ol
3-(2-chlorophenyl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}propanamide
({4-ethyl-5-[1-(quinolin-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-(4-acetyl-1,4-diazepan-1-yl)-2-[3-(butylcarbamoyl)phenyl]acetic acid
6-[3-(2-methylpropyl)morpholine-4-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methoxy-5-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}phenol
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
3,3,3-trifluoro-1-{4-[4-(2-hydroxypropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propan-1-one
(3R,9R)-11-{[3-(methylsulfanyl)phenyl]methyl}-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazine
8-(2,3-dimethoxybenzoyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-methyl-4-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}piperazine-2-carboxylic acid
1-(cyclohexylmethyl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
3-[(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridin-2-amine
(2S,4R)-4-amino-1-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
N-methyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(oxolan-2-ylmethyl)pyridin-2-amine
1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-4-(furan-2-carbonyl)-1,4-diazepane
N-methyl-N-(2-phenylethyl)-1-(quinolin-5-ylmethyl)piperidin-3-amine
(3S,4R)-4-(4-fluorophenyl)-1-{imidazo[1,2-a]pyridin-2-ylmethyl}pyrrolidine-3-carboxylic acid
1-(2-{[(2-phenylethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-{2-[(2S)-pyrrolidin-2-yl]ethyl}quinoxaline-6-carboxamide
4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]pyridazine
N-benzyl-1-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide