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3-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-[3-(piperidine-1-carbonyl)phenyl]urea
2-amino-4-(5-hydroxy-2-methoxyphenyl)-6-(1H-indol-3-yl)pyridine-3-carbonitrile
(1S,5R)-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2-{3-[3-(6-methoxypyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}ethyl)dimethylamine
3-{5-[(2,4-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
4-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-6-hydroxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
8-(2,3-dimethylbenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-[1-(furan-3-carbonyl)piperidin-2-yl]pyridine
(4-{[2-(3-fluoro-4-methylphenyl)-1H-imidazol-1-yl]methyl}phenyl)methanamine
(2R,6S)-4-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2,6-dimethylmorpholine
(1S,3R)-3-amino-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]cyclopentane-1-carboxamide
N-cyclopropyl-4-acetamido-N-{[3-(2-methylpropoxy)phenyl]methyl}benzamide
1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-2-(2-methyl-1H-imidazol-1-yl)propanamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4,4,4-trifluorobutanamide
2-(4-fluorophenyl)-N-{[(3S,4S)-3-hydroxy-1-(pyridine-2-carbonyl)piperidin-4-yl]methyl}acetamide
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-N,5-dimethyl-N-(2-phenylethyl)thieno[2,3-d]pyrimidine-6-carboxamide
(1R,5R)-N,N-dimethyl-6-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
methyl 7-oxo-3-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[3-(4-methanesulfonylphenyl)phenyl]-1-(prop-2-en-1-yl)-1H-pyrazole
1-benzyl-N3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(6-aminopyridine-3-carbonyl)-3-propylpiperidine-3-carboxylic acid
N,N-dimethyl-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine-1-sulfonamide
methyl 2-[(2,6-dihydroxyphenyl)formamido]-2-(3-methylphenyl)acetate
(3S)-3-(dimethylamino)-N-(4-phenylphenyl)pyrrolidine-1-carboxamide
4-benzyl-1-[3-(3-methoxyphenyl)propanoyl]-1,4-diazepan-5-one
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(cyclopropylmethyl)-2-[(1-ethyl-1H-indol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-3-acetyl-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-phenylpropanamide
N-(1-benzylpiperidin-3-yl)-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
5-(2-chlorophenyl)-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-ethoxyphenyl)ethan-1-one
3-({4-[5-chloro-2-(prop-2-en-1-yloxy)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-5-methyl-1,2,4-oxadiazole
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-(3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)-6-methoxypyrimidine
(4aS,8aR)-6-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
ethyl 4-{[3-(1H-pyrazol-5-yl)phenyl]carbamoyl}piperazine-1-carboxylate
(3R,9aR)-3-benzyl-8-(3-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2,2-diphenylethyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]morpholine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-ethyl-N,7,8-trimethyl-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]but-3-en-1-one
N-[(1S,2R)-2-aminocyclobutyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(4-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}-1,4-oxazepan-6-yl)methanol
methyl 2-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-5-methyl-1H-imidazole-4-carboxylate
4-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}pyrimidin-2-amine
N-methyl-N-(oxan-4-yl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(pyridin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one