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2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
2-(dimethylamino)-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
6-methyl-2-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
3-(2H-1,3-benzodioxol-5-yl)-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1-phenyl-1H-pyrazole
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(2S,4S)-1-[(2,5-dimethylphenyl)methyl]-N-ethyl-4-(furan-3-amido)pyrrolidine-2-carboxamide
[1-({[6-(propan-2-yl)pyrimidin-4-yl]amino}methyl)cyclopentyl]methanol
2-(ethoxymethyl)-N-[4-(furan-2-yl)phenyl]pyrrolidine-1-carboxamide
6-(isoquinolin-5-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(furan-3-carbonyl)piperazin-2-one
4-{[(2S)-1-methoxy-3-phenylpropan-2-yl]carbamoyl}-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
3-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2-methoxyquinoline
4-[3-(benzyloxy)azetidine-1-carbonyl]-2-(pyridin-4-yl)quinoline
5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
4-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}-2-phenyl-1,3-oxazole
1-(4-{4-[3-(diethylamino)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)-3-methoxypropan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]acetamide
(2E)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-3-phenylprop-2-enamide
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]pyridine-4-carboxamide
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-1-(2-methoxyacetyl)piperidine-4-carboxamide
6-(2-fluorophenyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}imidazo[2,1-b][1,3]thiazole
N'-methyl-N-(5-methyl-1,2-oxazol-3-yl)-N'-{[2-(2-methylpropoxy)phenyl]methyl}ethanediamide
2-[(4-chlorophenyl)amino]-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
(3S)-4-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-3-ethylmorpholine
(2S)-2-[(6-methyl-2-phenylpyrimidin-4-yl)amino]-2-phenylethan-1-ol
N-(3-methoxypropyl)-N-[(4-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
1-[(4aR,8aS)-1-(1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-methoxyethan-1-one
2-phenyl-1-[4-(3-phenylprop-2-yn-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
(2S,4S,5R)-4-[(carboxymethyl)(methyl)carbamoyl]-5-(2-chlorophenyl)-1,2-dimethylpyrrolidine-2-carboxylic acid
N-[2-(1H-indol-3-yl)ethyl]-6-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1'-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}azetidin-3-ol
(2R,3S,6R)-5-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)piperidine-1-carboxamide
4-(5-methylpyridin-2-yl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-ol
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(oxolane-2-carbonyl)piperazine
4-(1-ethyl-1H-imidazol-2-yl)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidine
2-ethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
(2S)-2-{[(4-hydroxyquinolin-2-yl)methyl]amino}-3-phenylpropanamide
1-{1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
(3R,9aR)-8-[(3,4-dimethylphenyl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(2H-1,3-benzodioxol-5-yl)-1-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-amine
(1S,2S)-2-[4-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperazin-1-yl]cyclohexan-1-ol
3-(5-fluoro-2-methylphenyl)-5-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,2,4-oxadiazole
N-[2-(pyrazin-2-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[3-(4-methyl-1,3-thiazol-5-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-(hydroxymethyl)-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]azepan-4-ol