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1-[(3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)methyl]-1H-pyrazole
1-[(3-chlorophenyl)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-4-(4-methylpiperazin-1-yl)-N-[1-(4-methylpyridin-2-yl)propan-2-yl]benzamide
1-(2-chloro-4-fluorobenzenesulfonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
ethyl 3-(2-phenylethyl)-1-(4,4,4-trifluorobutyl)piperidine-3-carboxylate
5-chloro-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
(1R,5S,6S)-6-({4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
2-(3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
1-methyl-N-[2-(4-methylbenzenesulfonyl)ethyl]azepane-2-carboxamide
4-{4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanoyl}piperazin-2-one
N-(1-phenyl-1H-pyrazol-5-yl)-2-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]acetamide
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclopropylacetamide
6-({[2-(diethylamino)pyridin-3-yl]methyl}amino)pyridine-2-carbonitrile
4-[(3S,5R)-5-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]piperidine-3-carbonyl]morpholine
N-methyl-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
1-(4-ethylpiperazin-1-yl)-3-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]propan-1-one
N-benzyl-1-[1-(3-methylbutanoyl)piperidin-4-yl]piperidine-3-carboxamide
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl][(2-fluorophenyl)methyl](2-methoxyethyl)amine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(pyridin-2-ylsulfanyl)acetamide
2-[1-(oxane-4-carbonyl)pyrrolidin-3-yl]benzoic acid
(3S,5S)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
N-(3-{[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methoxy}phenyl)propanamide
N-[2-chloro-5-(methylcarbamoyl)phenyl]-2-(pyridin-2-yl)piperidine-1-carboxamide
2-chloro-N-[2-(cyclopent-1-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]-1-(pyridin-4-ylmethyl)urea
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}propan-1-one
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl){[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
[(3-fluoro-2-methylphenyl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine
(1S,5R)-3-(oxan-4-yl)-6-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
3-methyl-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}pyridine-2-carboxamide
5-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-ethylpyrimidin-2-amine
3-[4-(3-chloro-4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
1-[2-(1H-imidazol-4-yl)ethyl]-4-(2-phenylethyl)-1H-1,2,3-triazole
(1R,9S)-5-amino-3-[(benzyloxy)methyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
7-[(2,3-dimethoxyphenyl)methyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole
(3S,7S,8aS)-7-[({3-[2-(dimethylamino)ethoxy]phenyl}methyl)amino]-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-chloro-4-fluoro-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-benzothiophene-2-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1,2-oxazolidin-2-yl)propanamide
2-[3-({[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]carbamoyl}amino)phenyl]-N-methylacetamide
benzyl[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
3-{methyl[2-(1,2,4-oxadiazol-3-yl)ethyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
5-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-[({1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
3-[2-(3-cyanophenyl)-1H-imidazol-1-yl]-4-methyl-N-(propan-2-yl)benzamide
N-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide