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2-{8-[3-(5-methylfuran-2-yl)butyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
N4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(morpholin-4-yl)propan-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
N,N,4-trimethyl-3-({[(1-propylcyclobutyl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(4-fluorophenyl)piperazin-2-one
2-(benzyloxy)-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-5-(3-methoxyphenyl)-1,2,4-triazine
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
5-(2-fluorophenyl)-4-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}-2-(pyridin-3-yl)pyrimidine
8-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-{4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2,4-dimethylbenzamide
5,6-dimethyl-2-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
4-(3-chloro-4-fluorobenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-ethyl-3-(2-methylpropyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazole-5-carboxamide
1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetamide
2-(3-methoxyphenyl)-N-(thiophen-3-ylmethyl)acetamide
(1R,5R)-3-methanesulfonyl-6-(5-phenyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-(pyridine-3-sulfonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(3-methoxyphenyl)ethyl]-N-methylbenzamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
(1S,2R)-N1-[2-(2-chlorophenyl)ethyl]-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
(furan-3-ylmethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amine
(4aS,7aR)-1-[3-(1H-imidazol-1-yl)propyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(cyclobutylmethyl)-3-(2-methyl-1-benzofuran-5-yl)-1-(oxolan-2-ylmethyl)urea
1-(6-cyanopyridin-2-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-amino-3-ethyl-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
3,4-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-5-sulfamoylbenzamide
N-{2-[2-(3,4-dichlorophenyl)-1H-imidazol-1-yl]ethyl}acetamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2R,6R)-4-(2-amino-6-methylpyrimidin-4-yl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-methyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-indole-6-carboxamide
1-[(2-chlorophenyl)methyl]-3-[(3-hydroxypiperidin-1-yl)methyl]-6-methyl-1,2-dihydroquinolin-2-one
3-[(2R,3R,6R)-5-(quinoxalin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1,2-dihydroquinolin-2-one
1-[(2-chloro-6-fluorophenyl)methyl]piperidine-3-carbonitrile
1-(2-methoxyethyl)-4-[7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
methyl (2S,4R)-4-hydroxy-1-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)pyrrolidine-2-carboxylate
2-(2-fluoro-6-methoxyphenyl)-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[(3S,4R)-1-(5-chlorothiophene-2-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-[(3R,4S)-1-[3-(dimethylsulfamoyl)propyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-{3-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]propyl}-2-methyl-1H-1,3-benzodiazole
N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-4-methyl-1,3-thiazole-5-carboxamide
2-{1-cyclopentyl-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol