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2-(5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl)pyridine
1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
2-[(4-chlorophenyl)methyl]-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}piperidin-2-one
N-(1H-indol-3-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
7-(2,2-dimethylpropyl)-2-(pyridin-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
7-(2-hydroxyethyl)-2-(5-methyl-2-phenylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-{4-[(2-aminopyrimidin-5-yl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-chloro-4-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
(1s,4s)-4-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
3-[3-(ethylsulfanyl)phenyl]-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
3-(5-tert-butyl-2-methoxyphenyl)-1-{2-[(pyridin-3-yl)amino]ethyl}urea
N-methyl-4-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridin-2-amine
N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-1-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
2-[4-(dipropylamino)piperidin-1-yl]-2-(4-fluoro-3-methylphenyl)acetic acid
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-(3-acetylphenyl)-3-(oxolan-3-ylmethyl)urea
1-(1,3-thiazol-2-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
N-cyclopropyl-4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperazine-2-carboxamide
2-[5-(2,6-difluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
4-[4-(2,6-dimethylquinoline-4-carbonyl)piperazin-1-yl]-6-methylpyrimidin-2-amine
1-ethyl-N-methyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-acetamidoethyl)piperidine-3,5-dicarboxamide
3-methyl-5-(2-propyl-1,3-thiazol-4-yl)-1H-1,2,4-triazole
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-(1-methyl-1H-1,3-benzodiazol-2-yl)benzamide
ethyl 3-[(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazol-4-yl)formamido]propanoate
2-{1-[(3-methylpyrazin-2-yl)methyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
5-[2-(piperidin-1-yl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[3-(3-fluorophenyl)phenyl]-1-[(2R)-pyrrolidine-2-carbonyl]piperidine-4-carboxamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chlorobenzamide
1-[(2,6-difluorophenyl)methyl]-3-(2-hydroxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
4-methyl-5-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,3-thiazole
7-(2-methylphenyl)-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(3-phenylpropyl)piperidin-3-yl]cyclopent-1-ene-1-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(trimethyl-1H-imidazol-2-yl)methyl]piperidine
1-[(4-chlorophenyl)methyl]-N-[(2,4-dihydroxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
2-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1,3-benzothiazole
(2S)-N-[1-(4-fluorophenyl)-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-(methylamino)propanamide
1-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}-3-methylbutan-1-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-(3,4-dichlorophenyl)-4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]morpholine
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-pentylpiperidine
1-methyl-4-(2-methylquinolin-6-yl)piperidin-4-ol
3-chloro-2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-6-methylpyrazolo[1,5-a]pyrimidine
5-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1,2-oxazole-3-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-(2-oxopyrrolidin-1-yl)butanamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(5Z)-2,4-dioxo-1,3-thiazolidin-5-ylidene]acetamide
methyl 4-methoxy-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]carbamoyl}amino)benzoate