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2-{[4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]acetamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-[(1,2-oxazol-3-ylmethyl)sulfamoyl]benzamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-oxopiperidin-1-yl)acetamide
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
1-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-3,3-dimethylurea
3-[1-(4-cyclopropanecarbonylphenyl)-1H-pyrazol-3-yl]pyridine
N-{1-[3-(piperidin-4-ylmethyl)benzoyl]piperidin-4-yl}acetamide
2-(1-methyl-1H-pyrazol-3-yl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(pyridin-2-ylmethyl)pyridin-2-amine
2-(4-methyl-1H-pyrrole-2-carbonyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(2-ethoxy-5-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}phenyl)methanol
3-(1-hydroxy-3-methylbutan-2-yl)-1-[6-(3-methoxyphenoxy)pyridin-3-yl]urea
(3S,4R)-1-[2-(3-fluorophenoxy)acetyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-methyl-5-{4-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
6-(2-chlorophenyl)-2-{4-[(2-methylpyrrolidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
(2S)-2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-2-phenylethan-1-ol
2-[4-(2-methoxyethoxy)phenyl]-2-[4-(4-methylphenyl)piperazin-1-yl]acetic acid
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-(pyrrolidin-1-ylmethyl)benzamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[(5,6-dimethylpyridin-3-yl)methyl]-4,6-dimethylpyrimidin-2-amine
2-(3-fluorophenyl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
5-(3-methoxyphenoxymethyl)-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-(3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-oxopropyl)-2-fluorobenzamide
2-cyclopropyl-N-[(1-methanesulfonylpiperidin-3-yl)methyl]pyrimidine-5-carboxamide
3-[(1S,2R)-2-aminocyclobutyl]-1-(3-chloro-2-methylphenyl)urea
2-methyl-N-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(oxane-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2,7-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]quinoline-4-carboxamide
(3R,4R)-4-ethyl-1-(thiophene-3-carbonyl)piperidine-3,4-diol
(1S,5R)-3-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-fluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
6-methyl-3-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
6-ethyl-N-[1-(1H-imidazol-2-yl)ethyl]-2-methylquinoline-4-carboxamide
3-(piperidin-1-ylmethyl)-1-[(5-propylfuran-2-yl)methyl]piperidine
N-(1,4-dioxan-2-ylmethyl)-3-{methyl[2-(methylsulfanyl)ethyl]sulfamoyl}benzamide
1-{4-[2-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}ethan-1-one
N-[2-(benzyloxy)ethyl]-1-(carbamoylmethyl)piperidine-4-carboxamide
3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(1,3,4-thiadiazol-2-yl)urea
N,1-dimethyl-2-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-dihydroquinoline-3-carboxamide
7-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
7-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(4aS,8aR)-1-butyl-6-[(4-oxo-4H-chromen-3-yl)methyl]-decahydro-1,6-naphthyridin-2-one
{7-[3-methyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
2-methyl-5-(2-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one