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N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
1-[2-(dimethylamino)ethyl]-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[3-(3-chlorophenyl)phenyl]-1-(2-methoxyethyl)piperidine-4-carboxamide
{4-[(2-chlorophenyl)methyl]-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl}methanol
2-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]-2,3-dihydro-1H-isoindole
7-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methoxypropan-1-one
ethyl 2-[(3S,4R)-3-acetamido-4-(4-methoxyphenyl)pyrrolidin-1-yl]-1,3-oxazole-4-carboxylate
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2-(1H-pyrazol-1-yl)benzamide
4-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methylpyrimidine
1-(5-cyanopyridin-2-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-({4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
5-{[(1-cyclopentylpiperidin-4-yl)methyl]amino}-1-(cyclopropylmethyl)azepan-2-one
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[2-(pyridin-4-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[3-(1H-imidazol-5-yl)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-{6-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
2-(3-chlorophenyl)-N-[(4-hydroxyazepan-4-yl)methyl]acetamide
(3S,5R)-1-(1H-imidazol-2-ylmethyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-methyl-5-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,3-thiazol-2-amine
8-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decane
ethyl 4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
3-(4-acetylphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
1-(5-fluoro-1H-indole-2-carbonyl)-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4-diazepan-5-one
3-{[(2,6-difluorophenyl)methyl]amino}-N-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-sulfonyl)benzamide
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-2-(2-ethylpyrimidin-5-yl)quinoline
(1S,4S)-5-[(2S)-2-hydroxypropanoyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}piperidin-3-yl)benzoic acid
2-cyclobutyl-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-[(diethylamino)methyl]-5-ethyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
2-(3-hydroxypropyl)-8-[(4-methoxy-3-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(4-fluorophenyl)-2-hydroxyethyl]benzamide
N-(naphthalen-1-ylmethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-1-(3-chloro-1H-indole-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-(1-benzothiophen-5-ylmethyl)-1-(carbamoylmethyl)piperidine-4-carboxamide
4-(cyclopropanesulfonyl)-2-(6-methoxynaphthalen-2-yl)morpholine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
8-cyclopropanecarbonyl-2-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[3-(4-fluorophenyl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
(3S,9aR)-8-(3,5-dichlorobenzoyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)acetamide
N,N-dimethyl-3-{[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}benzamide
4-[(4-fluorophenyl)methyl]-11-[(pyridin-3-ylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3aR,6aS)-5-{[4-(2-methylphenyl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
4-({2-[1-(ethanesulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(3R,4R)-1-[2-(dimethylamino)benzoyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
N,N-diethyl-1-(1-ethyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-amine
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(2-ethylphenoxy)azetidin-1-yl]ethan-1-one
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}azepan-4-ol