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N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)acetamide
(3S)-3-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}azepan-2-one
N-(2-methoxyethyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-(4-fluorophenyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
2-({4-[(3-methoxyphenyl)methyl]piperazin-1-yl}methyl)pyridine-3-carboxylic acid
N-[(3S,4R)-1-[(3-cyanophenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-(3-cyanothiophen-2-yl)-4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}benzamide
1-{1'-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-[4-(6-methyl-2-propylpyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
1-{2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyrrolidin-2-one
7-cyclopentyl-2-(morpholine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(4-cyano-2-ethylphenyl)-2-(3-methoxypropyl)piperidine-1-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-3-phenylpropanamide
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-propylfuran-2-carboxamide
6-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
2-[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-phenylacetamide
5-{1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazol-4-yl}-2-methoxypyridine
N-(3-hydroxypropyl)-1-(1-{[4-(2-methylphenyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
(1R,3S)-3-methoxy-7-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-7-azaspiro[3.5]nonan-1-ol
3-[5-chloro-4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-methyl-1H-pyrazol-3-yl]-5-methyl-1,2-oxazole
[(3S,5R)-5-[(dimethylamino)methyl]-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperidin-3-yl]methanol
(2S,4S)-N,N-diethyl-4-(2-methoxy-4-methylbenzamido)-1-methylpyrrolidine-2-carboxamide
[(3-cyclopropyl-1H-pyrazol-5-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
1-(2-methoxyphenyl)-5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1H-1,2,4-triazole
N-[1-(furan-2-carbonyl)piperidin-3-yl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
4-({[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]carbamoyl}amino)-N-ethyl-3-methylbenzamide
4-(pyrrolidin-1-yl)-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-2-amine
4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N-propylbenzamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
1-{1-[4-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}piperidin-4-ol
1-methyl-4-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
6-[(2-aminopyridin-3-yl)methyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
(3-{3-cyclopropyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}propyl)dimethylamine
N-[(3S,4R)-1-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-2-(trifluoromethyl)benzamide
5-amino-2-(2-methoxyphenyl)-1-methyl-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,3-benzodiazole-7-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)oxane-2-carboxamide
2-(3-ethoxy-5-fluorophenyl)-2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]acetic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(4-methylpiperazin-1-yl)propanamide
4-(5-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
N-[(3-fluoro-4-methylphenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-benzyl-3-{2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
4-(3-cyclopropyl-5-{[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]methyl}-1H-1,2,4-triazol-1-yl)-2-methylpyridine
2-[2-(morpholin-4-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
N'-cyclooctyl-N-(1H-imidazol-2-ylmethyl)butanediamide
2-{[(4-cyanopyridin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide