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1-[4-(dimethylamino)azepan-1-yl]-4-(naphthalen-1-yl)butane-1,4-dione
2-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)furan-3-carboxamide
5-methoxy-2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-4H-pyran-4-one
1-(4-methoxyphenyl)-3-methyl-4-[2-(methylamino)acetyl]piperazin-2-one
7-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-2-oxa-7-azaspiro[4.5]decane
(2R)-2-amino-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-methylpentan-1-one
4-[(3-fluorophenyl)methyl]-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole-3-carbonitrile
4-cyano-N-(1-phenylbutyl)benzamide
4-(ethanesulfonyl)-2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenol
methyl 5-oxo-5-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pentanoate
2-(3-methoxypropyl)-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-(1-methylpyrrolidin-3-yl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(3aR,6aR)-2-[(3,5-difluorophenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
N-{1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidin-4-yl}methanesulfonamide
(3R,5S)-N-(2-methylpropyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
5-(5-ethylfuran-2-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
(1R,5R)-6-(2-methoxyethyl)-3-[4-(5-methylfuran-2-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(1-methyl-1H-indol-5-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]-N-[4-(trifluoromethyl)phenyl]piperidine-1-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-(thiomorpholin-4-yl)propan-1-one
N-[(2-methoxyphenyl)methyl]-2-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}acetamide
5-(methanesulfonylmethyl)-2-(4-methoxy-3,5-dimethylphenyl)pyridine
3-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-2-yl}pyridine
4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]butanamide
3-(6-methoxypyridazin-3-yl)-5-methyl-1H-indole
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(2-methoxyethyl)piperazine
3-[(4aR,7aS)-4-(4-hydroxybenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[3-(2-hydroxyphenyl)propyl]propanamide
(1R,3S)-3-(2-hydroxyethoxy)-7-(5-methylthiophene-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methyl-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
(3S,4R)-4-(3-methoxyphenyl)-1-[3-(pyridin-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-3-methylbut-2-en-1-one
7-methoxy-3-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazol-2-yl]quinolin-2-ol
2-[2-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)-4-(pyridin-2-yl)phenoxy]acetic acid
2-(4-fluoro-3-methylbenzenesulfonamido)-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]acetamide
[(3R,4R)-1-[(3,4-dimethylphenyl)methyl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
1-({5-[1-(cyclopropylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)azepane
(3aR,6aR)-2-benzyl-5-(3-methylbut-2-enoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{1-[6-(1-hydroxyethyl)pyridin-2-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-{4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
(1R,5S,6S)-6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
methyl 6-[(2-ethyl-2-methyl-3-oxopiperazin-1-yl)methyl]pyridine-2-carboxylate
2-[(3-{[(5-fluoro-2-methylphenyl)methyl]carbamoyl}phenyl)amino]acetic acid
2-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1,4-diazepan-6-yl}acetic acid