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(2R,6R)-4-[3-(ethylsulfanyl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carboxamide
9-[2-(azepan-1-yl)acetyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-1,3-thiazole-4-carboxamide
(1S,5R)-3-[2-(benzenesulfonyl)ethyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-[3-(3,4-dimethoxyphenyl)propanoyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-methyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-[4-({3-[(3-fluorophenyl)amino]piperidin-1-yl}sulfonyl)phenyl]acetamide
5-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-4-methylpyrimidin-2-amine
9-(2-chloropyridine-4-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
[1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
1-(2,3-dihydro-1H-inden-2-yl)-4-(pyrazin-2-yl)-1,4-diazepane
5-[(cyclopropylmethyl)(propyl)amino]-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[5-(2-amino-2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]acetamide
2-[(3-chloro-4-hydroxyphenyl)methyl]-8-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{[(2-methoxyphenyl)methyl]amino}-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
8-(1-benzofuran-2-ylmethyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-N-(2-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)propanamide
1-({3-methoxy-4-[3-(trifluoromethyl)phenoxy]phenyl}methyl)pyrrolidine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(2S)-2-{[6-(methoxymethyl)pyrimidin-4-yl]amino}-4-methylpentanamide
4-[2-(1H-imidazol-2-yl)benzoyl]-3-propylmorpholine
(3aR,5R,6S,7aS)-2-({2-[3-(dimethylamino)propoxy]-3-methoxyphenyl}methyl)-octahydro-1H-isoindole-5,6-diol
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
5-methoxy-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
(2S,4R)-4-amino-1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2,5-dimethyl-3-[4-(1H-pyrazol-3-ylmethyl)piperazin-1-yl]pyrazine
5-methanesulfonyl-2-[(1-methylpiperidin-4-yl)methyl]-4-(piperidin-3-yl)pyrimidine
2-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
5-[2-(2-aminoethyl)morpholin-4-yl]-2-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
6-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-2-carbonitrile
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-fluorophenyl)methyl]-1,2-oxazole-3-carboxamide
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-4-(quinoxalin-6-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3,3-diphenylpiperidin-1-yl)propanamide
3-[3-(1,4-oxazepan-4-yl)propyl]-4,5,6,7-tetrahydro-2H-indazole
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-ethyl-3-(pyridin-2-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopentyl-4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[(1-hydroxycyclohexyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-2-yl}ethan-1-ol
2,4-dimethyl-N-(4-{4-[(pyridin-4-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
1-{2-[(1E)-3,3-dimethylbut-1-en-1-yl]pyridine-4-carbonyl}-4-methylpiperazine
4-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]phenol
4,6-dimethyl-1-{2-oxo-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2-dihydropyrimidin-2-one
1-(2-methylpropyl)-3,8-bis(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-methylpropanoyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-butanamido-N-methyl-N-[3-(oxolan-2-yl)propyl]benzamide