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7-fluoro-N-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-2-methylquinoline-4-carboxamide
N,N-diethyl-1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3-carboxamide
3-(pyrrolidin-1-ylmethyl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidin-3-ol
N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
3-[1-(1-benzofuran-2-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
2-(4-ethoxyphenyl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4-oxazepane
N-[2-(4-hydroxypiperidin-1-yl)ethyl]-3-methyl-5-propyl-1-benzofuran-2-carboxamide
6-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-(cyclopropylmethyl)-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-3-(propan-2-yl)-1,4-diazepan-5-one
(4aS,8aR)-6-(3-methoxypropyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(1-benzothiophen-2-ylmethyl)-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
[(3R,4R)-1-[(8-methoxyquinolin-2-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-[2-(methylsulfanyl)ethyl]piperazine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazole-3-carboxamide
N-cycloheptyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
8-[2-(4-hydroxyphenyl)acetyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
6-methyl-5-[5-(1-methyl-3-propyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
2-(methoxymethyl)-5-{[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyrimidine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(piperidin-4-yl)piperidine
7-(1-benzothiophen-3-yl)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,5R)-6-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-({5-[(2,3-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
(3R,4R)-1-[4-methoxy-3-(morpholin-4-yl)benzoyl]-3,4-dimethylpyrrolidin-3-ol
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
4-phenyl-3-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(pyridin-4-ylmethyl)piperidin-4-ol
2-cyclopentyl-N-[3-(4-{[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
4-methyl-2-(pyridin-3-yl)-6-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}pyrimidine
6-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylpyrazin-2-amine
4-hydroxy-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
6-fluoro-2-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]quinolin-4-ol
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(azocane-1-carbonyl)-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
2-[1-(6-methoxyquinolin-3-yl)-1H-pyrazol-4-yl]ethan-1-ol
8-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
4-(3-fluorophenoxy)-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid
6-methyl-14-(3-phenyl-1H-pyrazol-4-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(2R,3R)-3-amino-1'-(6-methyl-2-propylpyrimidin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[1-(2-phenylethyl)piperidin-3-yl]-3-(1H-pyrazol-1-yl)propanamide
2-[4-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)phenoxy]acetamide
5-{[4-(4-ethylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
[1-({methyl[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)cyclopentyl]methanol
2-benzyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3-thiazole-4-carboxamide
N-cyclopentyl-4-oxo-4-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]butanamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-3-yl]methanol
9-ethyl-1-methyl-4-(3-methylbenzenesulfonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-methyl-2-(1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)-1H-1,3-benzodiazole
methyl[(6-methylpyridin-2-yl)methyl][1-(pyrazin-2-yl)propan-2-yl]amine