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methyl 5-({[4-(2-hydroxyethoxy)phenyl]methyl}amino)-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
1-(4-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}thiophen-2-yl)ethan-1-one
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
7-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-phenoxypiperidine-4-carboxylic acid
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
2,2-dimethylpropyl 2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxylate
3-methyl-6-{5-[2-(propan-2-yl)-1,3-thiazol-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
3-(1H-imidazol-4-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(1H-pyrrol-1-yl)propan-1-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]morpholine-4-sulfonamide
(3S,5S)-1-benzyl-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
5-methyl-4-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-1-(4-methylphenyl)piperazin-2-one
9-(4-cyclopentylpyrimidin-2-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3-chlorophenyl)-4-[1-(3-methoxybenzoyl)piperidin-3-yl]piperazine
2-{[(butylcarbamoyl)methyl](methyl)amino}-2-(4-fluoro-3-methylphenyl)acetic acid
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methanol
6-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]ethan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
N-(4-fluoro-2-methylphenyl)-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]propanamide
(2R)-2-amino-3-(ethylsulfanyl)-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}propan-1-one
N-[(3S,4R)-1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-4-propylpyrrolidin-3-yl]methanesulfonamide
methyl (2S)-2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2-phenylacetate
N-[1-(dimethylsulfamoyl)azepan-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]pent-4-enamide
N-[2-(1-methyl-1H-pyrrol-2-yl)ethyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopropyl-4-methoxy-3-({1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-yl}oxy)benzamide
[2-(3-fluorophenyl)ethyl]({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
2-(4-fluorophenoxy)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]acetamide
N3-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-(propan-2-yl)-1H-pyrazol-1-yl]-4-(4-fluorophenyl)-5-methylpyrimidine
1-benzyl-4-[6-phenyl-2-(pyrrolidin-1-yl)pyridine-3-carbonyl]piperazine
N-(propan-2-yl)-4-{[3-(4H-1,2,4-triazol-4-yl)propyl]sulfamoyl}benzamide
3-cyclopropyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
5-(methoxymethyl)-N-(2,2,2-trifluoroethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]benzamide
1,9-dimethyl-4-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]-1,4,9-triazaspiro[5.5]undecane
2-{[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
1-{3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]propanoyl}-1,4-diazepan-5-one
N-[2-(dimethylamino)ethyl]-4-methoxy-3-{[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]oxy}benzamide
methyl 2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}piperidine-1-carboxylate
1-{3-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
(benzylsulfamoyl)({pyrazolo[1,5-a]pyridin-3-ylmethyl})amine
(1R,5S,8R)-N,N-dimethyl-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3-azabicyclo[3.2.1]octan-8-amine
2-({1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}amino)pyridine-3-carboxamide
methyl 4-[4-(2-{[(1-ethylpyrrolidin-2-yl)methyl]carbamoyl}ethyl)piperidin-1-yl]-4-oxobutanoate
1-[3-(5-methylfuran-2-yl)benzoyl]-4-[2-(pyrrolidin-1-yl)ethyl]piperazine