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(1R,3S)-3-ethoxy-7-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-[(1-methyl-5-phenyl-1H-pyrazol-3-yl)methyl]pyrimidin-2-amine
3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-5-(2-methylpropyl)-1,2-oxazole
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidin-3-yl]acetamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(2-oxopiperidin-1-yl)acetamide
3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-ylmethyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
2-(1H-imidazol-2-yl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]benzamide
1-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
N-(3-oxo-3-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propyl)methanesulfonamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine
N-(2,4-dimethoxyphenyl)-3-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}propanamide
2-amino-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-6-(2-methylpropyl)pyrimidine-4-carboxamide
2-(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
3-{3-[({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)methyl]-1H-indol-1-yl}propanamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
6-(2-aminoethyl)-N-methyl-N-(naphthalen-1-ylmethyl)pyrimidin-4-amine
2-(4-{[2-(2-phenylethoxy)phenyl]methyl}morpholin-3-yl)acetic acid
[(3R,4R)-1-(3-ethyl-1H-indole-2-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
propan-2-yl 2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carboxylate
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-methoxy-5-sulfamoylbenzamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl}pyridine
N-methyl-3-(methylsulfanyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
(2S,4R)-4-amino-N-methyl-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}pyrrolidine-2-carboxamide
cyclopentyl 4-(2-ethyl-4-methyl-1,3-oxazole-5-amido)benzoate
(3S,4R)-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
7-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1,3-dimethyl-6-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclopropanecarboxamide
N-cycloheptyl-1-cyclopropyl-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
1-{1-[1-(4-fluorophenyl)cyclopropanecarbonyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-chloro-5-(2,4,6-trimethylphenyl)pyrazine
2-methyl-N-({7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)butanamide
methyl 2-[(1,4-oxazepan-6-ylmethyl)amino]pyridine-3-carboxylate
2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[3-(pyridin-2-yl)propyl]acetamide
3-{[ethyl(methyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-cyclohexyl-N-methylpiperidine-4-carboxamide
2-(isoquinoline-1-carbonyl)-6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-2-(piperidin-1-yl)pyrimidine
N-[(2-chlorophenyl)methyl]-3-cyano-5-fluoro-N-(propan-2-yl)benzamide
4-{4-[2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)acetyl]piperazin-1-yl}benzonitrile
6-(azepan-1-yl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-cyclopropyl-3-({1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
(3S,4S)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(naphthalen-2-yl)piperidin-3-ol
4-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-2,6-dimethoxyphenol
3-chloro-N-methyl-N-{2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]ethyl}benzamide