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2,3-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}quinoxaline-6-carboxamide
2-(1-methylcyclopropanecarbonyl)-N-(oxolan-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-(5-fluoropyrimidin-2-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
3-(dimethyl-1,2-oxazol-4-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N'-cyclooctyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]butanediamide
1-methyl-2-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-imidazol-2-yl)-1H-1,3-benzodiazole
2-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
3-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-5-yl]-1-[2-(1H-pyrazol-1-yl)ethyl]urea
4-cyclobutyl-6-methyl-N-[1-(6-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
[(2-butyl-1H-imidazol-4-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-[(4-fluorophenyl)methyl]-4-({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amino)pyrrolidin-2-one
(2S)-2-({[7-chloro-2-(2-phenoxyethoxy)quinolin-3-yl]methyl}amino)-3-(1H-imidazol-4-yl)propan-1-ol
(4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)methanol
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
3-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}pyridin-2-amine
2-({[3-(dimethylamino)propyl](methyl)amino}methyl)-6-fluoroquinolin-4-ol
1-cyclohexyl-4-(1-ethyl-1H-pyrazole-4-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)methylamine
N-(4-{[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]methyl}phenyl)acetamide
2-{[(3S,4S)-4-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl]methyl}benzoic acid
1-(4-amino-5-methylpyrimidin-2-yl)-4-(1H-1,3-benzodiazol-1-yl)piperidine-4-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-methoxyphenyl)methyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2S,4R,6S)-2-(2-methoxypyrimidin-5-yl)-6-(2-phenylethyl)oxan-4-yl]acetamide
N-butyl-3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
5-[(furan-3-ylmethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
[2-(2-ethoxyphenoxy)ethyl][(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]methylamine
N,1-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-cyclohexyl-2-(9H-purin-6-yl)-2,7-diazaspiro[4.5]decan-6-one
methyl 6-(cyclopent-1-ene-1-carbonyl)-2-[(2,3-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-5-methyl-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]ethan-1-one
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine
(3aR,6aR)-2-[2-(methylsulfanyl)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-benzyl-N,1-dimethyl-5-{[2-(pyridin-3-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4-fluorophenyl)methyl]-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-[1-(cyclopent-3-ene-1-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine-3-carboxamide
3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-indazole
5-[2-(2-ethoxyethoxy)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(morpholin-2-ylmethyl)-6-phenylpyridazin-3-amine
2-(3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carbonitrile
3-(1H-pyrazol-4-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
4-(1-hydroxybutan-2-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
[4-(1,3-benzothiazole-6-carbonyl)-1,4-oxazepan-6-yl]methanol
1-(1-benzylpiperidin-4-yl)-N-[2-(furan-2-yl)ethyl]piperidine-3-carboxamide
N-benzyl-4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-sulfonamide
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(pyrrolidin-1-yl)propanamide