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N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(pyridin-4-yl)propanamide
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}pent-4-enamide
ethyl 4-[(4-{[1-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
4-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)amino]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
8-[(3-fluorophenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-(3,4-dimethoxybenzenesulfonyl)-8-methyl-2,8-diazaspiro[4.5]decane
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-[(4-methylpiperidin-1-yl)methyl]piperidin-2-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
7-(3-chlorophenyl)-4-(piperidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,2-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-ethyl-4-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
3-[3-(hydroxymethyl)phenyl]-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
6-chloro-2-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-imidazol-2-yl}quinoline
2-(4-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-pyrrole-3-carbonitrile
5-{4-[1-(dimethylamino)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl(3-methylbut-2-en-1-yl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(furan-2-yl)ethane-1,2-dione
1-{furo[3,2-c]pyridin-4-yl}-4-(pyridin-3-yl)piperidin-4-ol
[5-chloro-7-(1,2,3,4-tetrahydroisoquinolin-7-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[(1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
N-[(3S,4R)-1-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-2-yl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-{[3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-1-yl]methyl}phenol
N-[(3R,4S)-1-(2-methylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]cyclobutanecarboxamide
4-hydroxy-2-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
4-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]morpholine
1-[2-(3-fluorophenyl)ethyl]-N-methyl-6-oxo-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
5-{[4-(2-chloro-4-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-methyl-1H-imidazole
N,6-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-benzothiazol-2-amine
(3S)-3-benzyl-4-(1H-imidazol-2-ylmethyl)piperazin-2-one
3-[(2-fluorophenyl)formamido]-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)propanamide
4-[(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methyl]morpholine
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(pyridin-2-yl)propan-1-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-(furan-2-ylmethyl)piperidine-1-carboxamide
({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
6-[1-(5-hydroxypyrazine-2-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
(1R,3S)-3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]cyclopentan-1-amine
ethyl 1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
[(6-methoxypyridin-3-yl)methyl](3-phenylprop-2-yn-1-yl)propylamine
4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-[(3-methoxyphenyl)methyl]morpholine
6-[(propan-2-yl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-{4-[6-(2-methoxyphenyl)pyridazin-3-yl]phenyl}-2-methylpropanamide
(1R,5S,6R)-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-tert-butyl-2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
2-[5-(3,5-di-tert-butyl-4-hydroxyphenyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-3-yl]acetamide
5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-2-propyl-2,3-dihydro-1H-isoindole-1,3-dione