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1-(2,3-dimethyl-1H-indole-7-carbonyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
2,3-dimethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}quinoxaline-6-carboxamide
2-(1-methyl-1H-pyrrol-3-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
5-butyl-1'-(1-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[3-(1H-1,3-benzodiazol-1-yl)phenoxy]propanamide
(2R,6R)-10-methoxy-4-[3-(thiophen-2-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-(3-fluorophenyl)-4-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-2-one
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-6-methylpyridine-3-carboxamide
3-(1H-imidazol-2-yl)-N-[(5-methylpyrazin-2-yl)methyl]benzamide
5-(azepane-1-carbonyl)-N-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
N-[(2R)-2-hydroxypropyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
(1R,5S)-6-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-6-azabicyclo[3.2.1]octane
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(3-methylpiperidin-1-yl)propanamide
methyl 6-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyrazine-2-carboxylate
8-[(5-ethylfuran-2-yl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
8-(5-methyl-1,3-oxazole-4-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(2,6-dimethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}benzonitrile
7-(2,3-dimethoxyphenyl)-9-methoxy-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-(3-hydroxypropyl)-9-(2-methoxy-6-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N2,N2,5,6-tetramethyl-N4-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidine-2,4-diamine
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[4-(2-hydroxyethoxy)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-{3-[methyl(phenyl)amino]propyl}-1,1-dioxo-1λ6-thiolane-3-carboxamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
4-{[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
5-(4-fluorophenyl)-N-(thiolan-3-yl)pyrazolo[1,5-a]pyrimidin-7-amine
6-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
(1R,2S,9R)-11-[3-(trifluoromethyl)pyridin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
1-[(2,3-difluorophenyl)methyl]-3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
2-[5-(1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]benzonitrile
6-{1-[5-(morpholine-4-carbonyl)pyridin-2-yl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
5-methoxy-9-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
(2S,4S)-4-amino-1-{6-oxo-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraene-12-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 4-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}piperazine-1-carboxylate
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(4-hydroxyphenyl)methyl]acetamide
4-{[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
1-({5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
N-methyl-5-[(4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazol-1-yl)methyl]furan-2-carboxamide
(2R)-2-amino-N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]propanamide
2-{3-[(3-carbamoylphenyl)methyl]pyrrolidin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}butanamide
N,N-dimethyl-4-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)butanamide
7-[2-(1,3-thiazol-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]ethan-1-one
(3S,4R)-4-(4-fluorophenyl)-1-(pyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
methyl 2-(benzylsulfamoyl)-6-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methyl-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
1-{1-[(3,4-dimethoxypyridin-2-yl)methyl]piperidin-3-yl}-3-phenylpropan-1-one