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N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-1-(pyrrolidin-1-yl)cyclohexane-1-carboxamide
1-[2-(dimethylamino)-2-(3-methylphenyl)acetamido]cyclopentane-1-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(piperidin-1-yl)ethan-1-one
1-(1-ethylpyrrolidine-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
2-(1H-imidazol-1-yl)-1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-(4-{[1-(adamantan-1-yl)propyl]amino}piperidin-1-yl)ethan-1-one
N-[4-(4-methoxyphenyl)butan-2-yl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(piperidin-1-yl)benzamide
7-(3-methoxyphenyl)-2-(pyrimidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(5-methylfuran-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-oxoethyl)urea
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(4-propylmorpholin-2-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(methylsulfanyl)benzamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-[(2-fluorophenyl)methyl]-4-{4-[(5-methylthiophen-2-yl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl](2-phenylethyl)amine
(1S,5R)-3-(3,5-dimethyl-1-benzofuran-2-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(oxane-4-carbonyl)-4-(pyrazin-2-yl)-1,4-diazepan-6-ol
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[5-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-cyclobutyl-1-methyl-1H-1,3-benzodiazol-7-yl]oxolane-2-carboxamide
1-({4-[(1,2,3-thiadiazol-5-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
methyl (2S)-2-cyclopropyl-2-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamido]acetate
1-(4-{[(3-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-4-ol
4-{3-[1-(3,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]propyl}morpholine
6-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
2,6,8-trimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}quinoline-4-carboxamide
5-{[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
9-(cyclopropylmethyl)-4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,2-dimethyl-6-(propan-2-yl)pyrimidin-4-amine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine
4-(cyclohexylmethyl)-3-(1-ethyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
ethyl 1-{2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetyl}piperidine-4-carboxylate
1-[1-(5-amino-1H-pyrazole-3-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-fluorophenyl)-3-methyl-3-[2-(oxan-4-yl)ethyl]urea
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-3-fluoro-N-(pyridin-2-ylmethyl)benzamide
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-propanoyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one