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{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]methylamine
3-(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[2-(3-methoxyphenyl)piperidine-1-carbonyl]quinoxaline
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}furan-3-carboxamide
N-[(3R,4S)-1-[(3-methylpyrazin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
{3-[3-(1H-imidazol-2-yl)phenoxy]propyl}dimethylamine
5-(5-ethylpyrimidin-2-yl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-hydroxy-N-[3-(1H-indazol-1-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(4-fluorophenyl)oxane-4-carboxamide
(1R,2S,9R)-11-(3-fluoropyridin-4-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1,4-dithiepan-6-amine
5-benzyl-5-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-(1-benzofuran-2-ylmethyl)-1-(2-methoxyacetyl)piperidine-4-carboxamide
3-(1H-1,2,3,4-tetrazol-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
methyl 6-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}pyridine-2-carboxylate
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
1-[1-methyl-5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-1H-pyrrol-3-yl]ethan-1-one
(3R,5S)-N-(2-methylpropyl)-5-(morpholin-4-ylmethyl)-1-(2-phenylethyl)piperidine-3-carboxamide
1'-(2-amino-6-methoxypyrimidin-4-yl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
6-[(1,3-dihydroxypropan-2-yl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})[2-(pyridin-4-yl)ethyl]amine
1-(2-methoxyethyl)-4-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)pyrrolidin-2-one
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-cyclohexyl-1,3-benzoxazole-6-carboxamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,2-oxazole
N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[2-(4-fluorophenyl)ethyl]-4-[4-(pyrazine-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-{[methyl(oxan-2-ylmethyl)amino]methyl}phenoxy)acetic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide
2-(5-acetylthiophen-3-yl)-1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-cyclopropyl-N-(oxan-4-yl)-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}[2-(diethylamino)ethyl]ethylamine
1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}-4-(thiophen-2-yl)butan-1-one
1-[4-(2-fluoro-4-methanesulfonylphenyl)piperazin-1-yl]-2-(morpholin-3-yl)ethan-1-one
(2R)-2-amino-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N2-[2-(dimethylamino)ethyl]-N5-[(2R)-3-methylbutan-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2,5-dicarboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(4-ethylpiperazin-1-yl)pyrimidine
3-({4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyridin-2-amine
(1S,5R)-6-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-2,2-dimethyl-1-(thiophen-2-yl)cyclopropane-1-carboxamide
2-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1-oxaspiro[4.4]nonane-4-carboxamide
N-{[8-(pyrimidin-4-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-N-(1,3-thiazol-5-ylmethyl)cyclopropanamine
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}urea
N,6-dimethyl-2-(morpholin-4-yl)-N-(oxan-2-ylmethyl)pyrimidin-4-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,2-dimethyl-5-sulfamoylbenzamide
1-[4-(3-{[(1-benzothiophen-2-ylmethyl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
(1S,5R)-6-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
(2R)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}propanamide