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6-{[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-({1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2,7-dimethyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
1-[2-hydroxy-3-(2-methoxy-4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenoxy)propyl]piperidin-4-ol
(3S,9aR)-3-[(benzyloxy)methyl]-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{4-[(3-ethyl-4-methylpiperazin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
5-({3-[4-(3-methoxypropyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-2-methylpyridine
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
[(2S,6S)-11-methoxy-4-(4-methoxypyrimidin-2-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
2-amino-4-(5-methoxy-3-methyl-1H-indol-2-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1-[2-(morpholine-4-carbonyl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-(4,7-dimethylquinazolin-2-yl)-N-[3-(propan-2-yloxy)propyl]azepan-4-amine
1-(2-aminoethyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(4-methoxyphenyl)ethyl]-2-{2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}acetamide
N-[(2-chloro-4-fluorophenyl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
[(1,2-dimethyl-1H-imidazol-5-yl)methyl](methyl)[2-(pyridin-4-yl)ethyl]amine
2-methoxy-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,4-diazepane
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(3-methylpyridin-4-yl)methyl]pyridin-2-amine
N-(furan-3-ylmethyl)-2-(N-phenylmethanesulfonamido)propanamide
N-{[(2S,4S)-4-fluoro-1-[4-(1H-pyrazol-1-yl)benzenesulfonyl]pyrrolidin-2-yl]methyl}acetamide
5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
2-amino-6-(2-fluoro-4-hydroxyphenyl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-3-ol
N-butyl-1-ethyl-N-(furan-2-ylmethyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-cyclopropyl-4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyridine-2-carboxamide
N1-butyl-N2-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-1,2-dicarboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(5-methylfuran-2-yl)methyl]piperidine-2-carboxamide
10-[2-(furan-2-yl)azepane-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
5-benzyl-4-(3-hydroxypropanoyl)-1-(4-methylphenyl)piperazin-2-one
(1R,5R)-N,N-dimethyl-6-[2-(phenylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(1,4-diazepane-1-carbonyl)-N-(oxolan-3-yl)benzene-1-sulfonamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanamide
N2-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
7-(2-cyclopentyl-2-phenylacetyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
11-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-cyclobutyl-5-{1-[3-(pyrazin-2-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-ethyl-6-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]pyrimidine
5-[2-oxo-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethyl]imidazolidine-2,4-dione
2-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-N-propylaniline
1-benzyl-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
1-[2-methoxy-4-({[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-1H-1,3-benzodiazole
3-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-3-(piperidin-3-yl)benzamide
7,7-dimethyl-N-[(6-methylpyridin-2-yl)methyl]-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
2-methylpropyl 4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carboxylate