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2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
N-[(2R,4R,6S)-2-cyclohexyl-6-[2-methyl-1-(morpholin-4-yl)propan-2-yl]oxan-4-yl]acetamide
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methylpyridazine-4-carboxamide
N-methyl-N-(pyrazin-2-ylmethyl)quinoline-6-carboxamide
(1R,5R)-6-{[3-(methylsulfanyl)phenyl]methyl}-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-phenylbenzoyl)piperazine
N-methyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)-N-(2-phenylethyl)acetamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-methyl-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-(2-methylphenyl)piperazin-2-one
4-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-1,2-dimethylpiperazine
7-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3R,5S)-1-benzyl-N-(2-methylpropyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
N-[(3-methoxyphenyl)methyl]-2-methyl-N-(prop-2-en-1-yl)-1,8-naphthyridine-3-carboxamide
N'-[2-(2-ethoxyphenoxy)ethyl]-N'-methyl-N-(1,3,4-thiadiazol-2-yl)ethanediamide
3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
8-cyclopropanecarbonyl-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(2-fluorophenyl)methyl]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
3-(4-fluorophenyl)-4-[2-(2,2,6,6-tetramethylpiperidin-4-yl)acetyl]piperazin-2-one
8-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
3-(4-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}piperazin-1-yl)pyrazine-2-carbonitrile
{2-[4-(3-methylphenoxy)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
1-(4-{[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)pyrrolidine
9-cyclopropanecarbonyl-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(2-fluorophenyl)-5-(furan-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-cyclopropyl-5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
(2S,4S)-4-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-N-ethyl-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
5-methoxy-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4H-pyran-4-one
4-[4-(furan-2-carbonyl)piperazin-1-yl]-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-6-methylpyridine-3-carboxylic acid
4-[(1-benzyl-1H-pyrazol-4-yl)methyl]morpholine
4-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1-(2-phenylethyl)piperazin-2-one
N-[(3,4-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)thiophene-2-carboxamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]propan-1-one
3-(2-fluoro-6-methoxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
9-(5-fluoro-2-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(6-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyridin-3-yl)methyl]morpholine
N-benzyl-2-ethoxy-N-(1,3-thiazol-2-ylmethyl)acetamide
1-(3-methoxypyrazin-2-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-(4-methoxy-3,5-dimethylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
2-[(3-methoxyphenyl)methyl]-8-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4-[3-(2-ethylphenoxy)azetidin-1-yl]-6-methoxypyrimidin-2-amine
9-(2,3-dihydro-1H-inden-1-yloxy)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-phenylpyrrolidin-3-ol