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2-[5-(5-hydroxypyrazin-2-yl)-3-phenyl-1H-1,2,4-triazol-1-yl]acetic acid
N-benzyl-2-(cyclopentylmethyl)-N,6-dimethyl-4-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-dihydropyridine-3-carboxamide
2-tert-butyl-6-(2,4,5-trimethylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-[2-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1H-imidazol-1-yl]-2,3-dihydro-1λ6-thiophene-1,1-dione
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
N-cyclohexyl-4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-1-carboxamide
N-[5-(cyclopropylcarbamoyl)-2-methoxyphenyl]-2-(4-fluorophenyl)azetidine-1-carboxamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
5-{1-[(2,4-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
(5S)-5-[({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
methyl 5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxylate
N-[(3S,4R)-1-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-amino-3-ethyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-hydroxy-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
3-({3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-{5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-ethyl-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-methylpiperidine-3-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-{2-[4-(3-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
4-({5-[1-(heptan-4-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine
2-{4-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)phenol
N3-{[3-(benzyloxy)phenyl]methyl}piperidine-1,3-dicarboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-N-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridine-6-carboxamide
ethyl 2-{1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperidin-2-yl}acetate
1-{2-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]pyrimidin-4-yl}piperidin-4-ol
(1R,5S,6R,7S)-3-(2-aminoethyl)-4-oxo-N-[2-(phenylsulfanyl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-4,6-dihydroxypyridine-3-carboxamide
N-(3-fluorophenyl)-3-{[3-(N-methylacetamido)pyrrolidin-1-yl]methyl}benzamide
N-[2-(2-hydroxyethoxy)ethyl]-1-benzothiophene-5-carboxamide
N4-[3-(1H-1,3-benzodiazol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-4-ol
1-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-[4-(pyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
(3S,4R)-4-(4-fluorophenyl)-1-{2-[(furan-2-ylmethyl)carbamoyl]ethyl}pyrrolidine-3-carboxylic acid
(2S,4S)-4-amino-N-ethyl-1-(5-ethyl-2-methylpyrimidin-4-yl)pyrrolidine-2-carboxamide
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
N-{[5-(quinolin-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
2-[5-(thiophen-2-yl)thiophen-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}pent-4-enamide
1-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
2-methyl-5-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
4-(1-methoxypropan-2-yl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
3-{[7-acetyl-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}propanamide
N-cycloheptyl-1-cyclopropyl-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(3-methoxypropyl)-8-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one