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N-(dimethyl-1H-1,2,4-triazol-3-yl)-2-(3-methoxyphenyl)piperidine-1-carboxamide
4-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]naphthalene-1-carboxamide
1-cycloheptyl-6-oxo-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
N-benzyl-1-[1-(2-hydroxyacetyl)piperidin-4-yl]piperidine-3-carboxamide
2-methyl-6-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-4-yl)pyrimidin-4-ol
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(ethylsulfanyl)propan-1-one
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]pyridine-4-carboxamide
N-{[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl}pyrazine-2-carboxamide
9-(3-methanesulfonylpropanoyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
4-(2-methoxyphenoxy)-1-[(3E)-pent-3-enoyl]piperidine-4-carboxylic acid
1-{2-[1-(2-methylphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}phenoxymethyl)pyridine
N-(2-{[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}quinolin-5-yl)acetamide
N-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-ethyloxan-4-amine
8-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
N-[2-fluoro-6-(trifluoromethyl)phenyl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
1-(2-ethoxyethyl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-[(3R,4S)-1-[(3-chloro-4-fluorophenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(3R,4R)-4-ethyl-1-(2-ethylpyridine-4-carbonyl)piperidine-3,4-diol
N-(3-benzamido-4-methoxyphenyl)-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-cyclopentyl-2-phenylethan-1-one
(2S)-N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-acetamido-4-(methylsulfanyl)butanamide
7-[(2-fluorophenyl)methyl]-2-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
(1S,5R)-6-benzyl-3-[4-(hydroxymethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methoxy-N-{4-methyl-3-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}carbamoyl)amino]phenyl}acetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(2-methoxyacetyl)-N-methylpiperidine-4-carboxamide
2-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-4-methylpyrimidine
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}[3-(4-fluorophenoxy)propyl]methylamine
1-[4-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
2-{methyl[(3-methylpyridin-2-yl)methyl]amino}-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
8-[(3,4-dimethoxypyridin-2-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
(2S,4R)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
(1S,6R)-3-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
4-methoxy-6-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
2-methyl-5-[4-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
1-[3-(2-chlorophenoxy)azetidin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
1-{2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]pyrimidin-4-yl}piperidin-3-ol
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-(3-phenylpropyl)benzamide
2-[4-(5-fluoropyrimidin-2-yl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-4-(morpholin-4-yl)-N-(pyridin-3-ylmethyl)benzamide
2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
(2R,6R)-4-[2-(4-methoxyphenyl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]azepane
1-{[3-(azocane-1-carbonyl)-1H-pyrazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole
2-(carbamoylamino)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide