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2,5-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazole
5-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-(4-methyl-1H-pyrazol-1-yl)-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[(2,4-dimethoxyphenyl)methyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-{2-oxo-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
8-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
8-methyl-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
N-[(6-hydroxypyrimidin-4-yl)methyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
2-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
5-butyl-N4,6-dimethyl-N4-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
(1R,3S)-3-(2-aminoethoxy)-7-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
(2S,4R)-N,N-diethyl-4-(2-hydroxyacetamido)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
N-methyl-2-phenyl-2-[(pyrimidin-2-yl)amino]acetamide
1-{3-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}pyrrolidin-2-one
7-(2,4-dimethoxybenzenesulfonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)pyrrolidin-2-one
1-(butan-2-yl)-N3-ethyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-[furan-2-yl(phenyl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-(1,4-dioxan-2-ylmethyl)-3-(oxan-4-yl)-5-(1H-pyrazol-3-yl)-1H-1,2,4-triazole
4-hydroxy-2-phenyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
3-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[3-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-methylpyridine-3-carboxamide
7-[(3-methoxyphenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{1-[4-(3-chlorophenyl)-5-[(cyclohexylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-5-(methoxymethyl)furan-2-carboxamide
1-(furan-2-ylmethyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]piperidine-4-carboxamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidine
ethyl 1-(3-chlorobenzenesulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
4-[2-(2-hydroxyethoxy)ethyl]-N-(4-methyl-2-oxo-2H-chromen-7-yl)piperazine-1-carboxamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
[(2-chloro-4,5-dimethoxyphenyl)methyl](methyl)(oxan-2-ylmethyl)amine
2-({2-[2-(propan-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}methyl)pyridine
8-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-(2-methoxyphenyl)propan-1-one
2-methyl-6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
1-{2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-methoxypropyl)-1-[2-(1-methyl-1H-indol-3-yl)acetyl]piperidine-3-carboxylic acid
3-[5-(4-methyl-1,3-oxazol-5-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
8-(1,3-benzoxazol-2-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
(1s,4s)-4-hydroxy-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}cyclohexane-1-carboxamide