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1-[(4-fluorophenyl)methyl]-4-{[5-(trifluoromethyl)pyridin-2-yl]amino}pyrrolidin-2-one
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
3-(2,4-dimethylphenyl)-1-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methylurea
3-[2-(7-methoxy-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]oxy}-3-chloro-N-(2-methoxyethyl)benzamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(cyclopropylmethyl)-N-propylacetamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(2S,4R)-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
N-[(2-chlorophenyl)methyl]-2-(2-oxopyrrolidin-1-yl)-N-(prop-2-en-1-yl)propanamide
1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-3-methylquinoxaline
4-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-(2-ethoxyethyl)-5-(4-propylpiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(3S,4R)-4-(4-methylphenyl)-1-(2-methylpropyl)pyrrolidin-3-yl]cyclopropanecarboxamide
3-[(3R,4S)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-[2-(methoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-(dimethylamino)-N-methyl-2-(2-methylphenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
3-{5-[3-(1H-pyrazol-4-yl)phenyl]-1,2,4-oxadiazol-3-yl}pyridine
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(2-phenylethyl)piperidine-4-carboxylic acid
(3S,4R)-3-(dimethylamino)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidine-1-sulfonamide
3-(benzyloxy)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
4-ethyl-3-[1-(pyrrolidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-N-(3-methyl-4-pentanamidophenyl)-3-propyl-1H-pyrazole-5-carboxamide
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
N-[2-(ethanesulfonyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-methylazepane-2-carboxamide
3-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]piperidine-1-carboxamide
3-(4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}-6-methylpyridine-3-carboxamide
2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2-methylpropan-1-ol
methyl (1R,3S,3aR,6aS)-1-ethyl-3-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)acetamide
N-(2,3-dihydro-1H-inden-5-yl)-4-(furan-3-carbonyl)-1,4-diazepane-1-carboxamide
N-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
2-[5-oxo-2-(thiophen-2-yl)cyclopent-1-en-1-yl]-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyridine
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-4-methoxy-3-methylbenzamide
1-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazole-5-carbonyl}-3-propylpiperidine-3-carboxylic acid
N-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-(3-methoxyphenyl)-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1H-pyrazole-4-carboxamide
2-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[1-(2-fluorophenyl)piperidin-4-yl]acetamide
1-[(2S,4R)-1-[(3-phenoxyphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
N-[(5-chloro-2-methoxyphenyl)methyl]-2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-ethylacetamide
2-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}quinoxaline