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3-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]benzonitrile
3-methyl-5-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazol-5-yl]-1H-1,2,4-triazole
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-[3-(pyridin-3-yloxy)propyl]acetamide
5-(3-fluoro-2-methylphenyl)-3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(oxan-4-ylmethyl)acetamide
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-cyclopropyl-1H-pyrazole-5-carboxamide
N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-amine
1-{2-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
ethyl 1-[2-(4-propanoylphenoxy)acetyl]piperidine-2-carboxylate
(2-chlorophenyl)methyl 3-aminoazepane-1-carboxylate
4,6-dimethyl-N,N-bis(2-methylpropyl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-chloro-N-{2-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
4-hydroxy-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-2-phenylpyrimidine-5-carboxamide
1-(benzenesulfonyl)-N-(1-phenoxypropan-2-yl)piperidin-4-amine
N,N-dimethyl-3-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-1H-1,2,4-triazol-5-amine
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]butan-1-one
6-[(4-ethoxyphenyl)methyl]-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-4-(pyrrolidin-1-yl)benzamide
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
2-{2-[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazine
propan-2-yl 4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
2-(3-hydroxypropyl)-9-[2-(1H-imidazol-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(2-methoxyphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
N-methyl-N-(oxolan-3-yl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[(3S)-3-ethylmorpholin-4-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}-N-methylethane-1-sulfonamide
1-ethyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-ethylpyrrolidine-2-carboxamide
4-(methoxymethyl)-5-methyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2-oxazole
1-[1'-(3-fluoro-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
8-(5-chloropyridine-3-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[1-(3-hydroxypyridine-2-carbonyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-{2-[(2-amino-6-methylpyrimidin-4-yl)amino]ethyl}-6-phenyl-2,3-dihydropyridazin-3-one
2-({[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}amino)pyridine-3-carboxamide
3-{[1-(2,3-dihydro-1H-inden-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
N,5,6-trimethyl-N-[(3-methylpyridin-4-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
N-[(4-fluorophenyl)methyl]-3-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
2-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-1,3-thiazole-4-carboxamide
2-{[(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)carbamoyl]amino}acetamide
2-[(2-methoxyethyl)(methyl)amino]-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-({[(2-aminopyridin-3-yl)methyl]amino}methyl)-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(2-hydroxyethyl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
methyl 6-[(4-methoxyphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[3-(1H-indol-1-yl)propyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
4-[(3-acetamidopyrrolidin-1-yl)sulfonyl]-N-(2-hydroxyethyl)benzamide
1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[4-(methylamino)pyrimidin-2-yl]piperazin-2-yl}ethan-1-ol