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2-methoxy-1-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)butan-1-one
(4S,4aS,8aS)-4-phenyl-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-decahydroquinolin-4-ol
2-(2-{[2-(4-ethoxyphenyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
methyl 1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
N-benzyl-N-ethyl-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
4-phenyl-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-4-(1H-pyrazol-4-yl)butan-1-one
8-chloro-3-[5-chloro-2-(propan-2-yloxy)phenyl]-[1,2,4]triazolo[4,3-a]pyridine
(3S,4S)-4-(4-fluorophenyl)-1-(2,2,6,6-tetramethylpiperidin-4-yl)piperidin-3-ol
6-[4-(cyclopropylmethyl)piperazin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-tert-butyl-6-{spiro[2.3]hexane-1-carbonyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-(1,3-benzoxazol-2-yl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-[(3-hydroxyphenyl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
[(3R,4R)-1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
6-fluoro-2-oxo-N-{3-[(pyridin-3-yl)amino]propyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
(2S)-N2-butyl-N2-(thiophen-3-ylmethyl)pyrrolidine-1,2-dicarboxamide
4-hydroxy-1-[4-(trifluoromethyl)benzoyl]piperidine-4-carboxylic acid
2-[4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]-1,3-benzoxazole
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-butoxyacetamide
1-[2-(5-{[(2-methylphenyl)amino]methyl}-1,2,4-oxadiazol-3-yl)ethyl]pyrrolidin-2-one
N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-{2-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(3-phenylpiperidin-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
3-(morpholin-4-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-cyclopropyl-5-(2-phenylbenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(4-methylpiperazine-1-carbonyl)-1-(2-propylpyridine-4-carbonyl)piperazine
5-(5-ethylfuran-2-yl)-4-phenyl-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
N-{[4-(2-methoxyethoxy)phenyl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyrimidin-4-ylmethyl)acetamide
2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}-2-[2-(methylsulfanyl)phenyl]acetic acid
4-{5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-sulfonyl]thiophen-2-yl}-2-methyl-1,3-thiazole
N-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]-3-[(thiophen-2-ylmethyl)amino]benzamide
N-[2-(3-fluorophenyl)ethyl]-5-{4-hydroxy-1-[(3-methylphenyl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
methyl 4-{2-[(1-benzylpyrrolidin-3-yl)carbamoyl]ethyl}piperidine-1-carboxylate
1-(3-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}phenyl)ethan-1-one
N,N-dimethyl-4-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperazine-1-carboxamide
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-ethoxypropan-1-one
4-chloro-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-(2-methoxyethyl)-8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-[2-(methylsulfanyl)pyrimidin-4-yl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[benzyl(methyl)amino]-3-[4-({[(6-methylpyridin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
6-[(3S)-3-ethylmorpholine-4-carbonyl]-1H-indole
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(4-methylpiperidin-1-yl)acetamide
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-{4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]phenoxy}acetamide
3-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline
2-{[5-fluoro-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethan-1-ol