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7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane
1-(3-{[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}propyl)piperidin-3-ol
N-[1-(4-hydroxyphenyl)-2-methylpropan-2-yl]-2-methyl-1,3-thiazole-4-carboxamide
2-(3-methylphenyl)-5-{[4-(thian-4-yl)piperazin-1-yl]methyl}pyrimidine
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
(1S,5R)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-{10,10-dichlorotricyclo[7.1.0.04,6]decan-5-yl}-3-methyl-1,2,4-oxadiazole
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
10-(3-hydroxypiperidine-1-carbonyl)-9-methoxy-3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-{3-oxo-3-[4-(pyridin-4-yl)piperidin-1-yl]propyl}azepan-2-one
{3-[(2,4-difluorophenyl)methyl]-1-(pyridin-4-ylmethyl)piperidin-3-yl}methanol
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]acetamide
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
8-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
1-[(4aR,8aS)-1-(2-fluorobenzoyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
N-{4-[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]phenyl}acetamide
1-(2-ethoxyethyl)-N-[(1-hydroxycyclohexyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
N-(3-methyl-1-propyl-1H-pyrazol-5-yl)-3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]benzamide
4-(4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanoyl)-1λ6-thiomorpholine-1,1-dione
1-[4-(furan-2-yl)phenyl]-N-[4-(methylamino)butyl]piperidin-4-amine
2-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)-5-fluoro-1-methyl-1H-indole
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(4-chloro-1H-pyrazol-1-yl)acetamide
3-[(3R,4S)-1-(1-benzofuran-5-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
8-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-8-chloroquinoline-2-carboxamide
1-(4-methyl-1,3-thiazol-2-yl)-4-(2-phenoxyethyl)piperazine
1,3-dimethyl-6-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
2-[(cyclopropylmethyl)sulfanyl]-1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]ethan-1-one
3-[(2-fluorophenyl)methyl]-4-[(2R)-3-methylbutan-2-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
5-[(adamantan-1-ylmethyl)(methyl)amino]-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
5-{[2-(diethylamino)ethyl](methyl)amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,4R)-4-cyclobutyl-3-methyl-1-{[3-(morpholin-4-yl)phenyl]methyl}piperidin-4-ol
4-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-1-(1H-indazol-5-yl)piperazin-2-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-5-phenyl-1H-pyrrole-2-carboxamide
methyl 2-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-1,3-oxazole-4-carboxylate
(2R,6R)-4-[2-(methylamino)-1,3-thiazole-4-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-4-(1H-pyrazol-3-yl)benzamide
7-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methoxy]-6-methyl-1H,2H,3H,4H-cyclopenta[c]chromen-4-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(furan-2-yl)-2-oxoacetamide
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(4-fluorophenyl)morpholine
5-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methyl-1,3-thiazole
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
3-methyl-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-{[2-(trifluoromethoxy)phenyl]methyl}urea