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2,3,6-trimethyl-4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]quinoline
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2,2-dimethylpropan-1-one
(3R)-N-benzyl-3-hydroxy-N,3,4,4-tetramethylpyrrolidine-1-sulfonamide
3-butyl-1-methyl-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
5-{3-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyrrolidin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-(furan-2-ylmethyl)-2-hydroxy-N-(1-hydroxybutan-2-yl)-5-(1H-pyrrol-1-yl)benzamide
N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[(4-chlorophenyl)methyl]-4-(5-ethyl-1,3-oxazole-4-carbonyl)piperazine
1-ethyl-4-{[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl}piperazine
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-N-(3-chloro-4-fluorophenyl)propanamide
2-acetyl-8-[(2-aminopyridin-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(1H-pyrazol-1-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidine-4-carboxylic acid
1-[(2S)-2-(3-benzyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]ethan-1-one
(3S,4R)-4-(3-fluorophenyl)-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrrolidine-3-carboxylic acid
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1-methylpiperidin-4-yl)piperidin-2-one
1-(3-methoxybenzoyl)-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
5-ethyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1,3-oxazole-4-carboxamide
1-[(1R,5R)-6-[(2,6-dimethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[2-(3-fluorophenyl)ethyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
5-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
N-[phenyl(pyridin-4-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-cyclopropyl-2-ethyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}butanamide
2-[4-(3,5-dimethylbenzoyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-methylthieno[2,3-d]pyrimidin-4-amine
15-methyl-13-oxo-N-[2-(pyridin-3-yl)ethyl]-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
4-methoxy-N-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[(4-acetylmorpholin-2-yl)methyl]-2-methylfuran-3-carboxamide
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-[4-(hydroxymethyl)phenyl]ethan-1-one
1-(2,4-dimethoxyphenyl)-3-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]urea
4-(piperidin-1-yl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine-4-carboxamide
4-hydroxy-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
(4aR,7aS)-1-(2-methoxyethyl)-4-[3-(pyridin-4-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[5-(4-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]phenyl}ethan-1-ol
(2E)-3-(3-fluorophenyl)-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
ethyl 2-[({2-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)(methyl)amino]acetate
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2H-1,3-benzodioxole-5-carboxamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-pyrazole-5-carboxamide
N2,N2-dimethyl-N4-{[1-(phenoxymethyl)cyclopropyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-hydroxy-N-methyl-N-(quinolin-5-ylmethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(1R,5R)-6-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-methyl-6-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-cyclopentyl-5-[4-(4-methylphenyl)piperazine-1-carbonyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
1,5-dimethyl-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1H-pyrazole-3-carboxamide
(3R,5S)-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-(4-{[methyl({[1-(morpholin-4-yl)cyclohexyl]methyl})amino]methyl}thiophen-2-yl)ethan-1-one
3-benzyl-4-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one