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(1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol
6-methyl-2-[3-(3-methylphenoxy)azetidin-1-yl]pyridine-3-carboxylic acid
1-methyl-4-[({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]piperidin-4-ol
2-(dimethyl-1,2-oxazol-4-yl)-N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(2S,4S)-4-amino-N,N-diethyl-1-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidine-2-carboxamide
2-(2-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrrol-1-yl)-1,3-thiazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-imidazol-2-ylmethyl)piperidin-3-ol
{3-[(3-methoxyphenyl)methyl]-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl}methanol
1-(2H-1,3-benzodioxol-5-yl)-N-[2-methoxy-2-(thiophen-2-yl)ethyl]piperidin-4-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[3-(4H-1,2,4-triazol-4-yl)phenyl]piperidine-1-carboxamide
1-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-(2-oxoazonan-1-yl)acetamide
6-cyclopentyl-N,1-dimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(azepan-1-yl)-3-[3-({[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}methyl)phenoxy]propan-2-ol
1-{1'-[(2,2-dimethyloxan-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-2-(2-hydroxyphenoxy)acetamide
N-methyl-5-[1-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
2-(2-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole
3-ethyl-5-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1,2-oxazole-4-carboxamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(naphthalen-2-yloxy)ethan-1-one
(1S,5R)-1,3,3-trimethyl-6-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-6-azabicyclo[3.2.1]octane
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
5-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-cyclopentyl-1H-imidazole
1-[(3-methoxyphenyl)methyl]-4-(pyrazin-2-yl)piperazin-2-one
7-(cyclobutylmethyl)-2-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(1H-pyrazol-3-yl)piperidine
3-(2-fluorophenyl)-3-phenyl-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
1-cyclohexyl-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
3-methyl-8-(quinoxaline-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-tert-butyl-4-{[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}furan-2-carboxamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-methyl-3-[3-(piperazin-1-yl)phenyl]-1H-indole
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(morpholine-4-carbonyl)-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline
(2E)-1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
2,3-dimethyl-7-[2-(methylamino)pyridine-4-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azetidin-3-yl}piperidine
4-(4-chlorophenoxy)-N,N-dimethylpiperidine-4-carboxamide
1-ethyl-N-[2-(4-methoxyphenyl)ethyl]-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]pyridazine