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1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-4-phenylpiperazine
N-(1-{[(1R,5S,6R)-3-(furan-2-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}piperidin-4-yl)pyrimidin-2-amine
1-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
7-(2,6-dimethylhept-5-en-1-yl)-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-(4-benzoylpiperazine-1-carbonyl)-2-(pyridin-2-yl)pyrimidin-4-ol
8-(2,6-dimethylpyrimidine-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{2-[(2-ethylphenyl)carbamoyl]ethyl}-5-oxopyrrolidine-3-carboxylic acid
1-(furan-3-carbonyl)-4-[4-(pyridin-3-yl)pyrimidin-2-yl]-1,4-diazepane
(4aS,7aR)-1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-{[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
(4aS,7aR)-1-(2-methylfuran-3-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{3-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-[4-(6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]acetamide
4-benzyl-1-[2-oxo-2-(piperazin-1-yl)ethyl]pyrrolidin-2-one
8-fluoro-4-oxo-N-[(4-sulfamoylphenyl)methyl]-1,4-dihydroquinoline-3-carboxamide
2-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}benzoic acid
1-(2-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
1-ethyl-N-[(2-methylphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(4-methoxybenzenesulfonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(1H-indole-2-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-{2-[2-(2-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}acetamide
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(1-benzofuran-2-ylmethyl)piperazine-2-carbonyl]-4-methylpiperazine
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
2-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
{1-[4-(trifluoromethoxy)benzenesulfonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
3-hydroxy-3-{[methyl(2-phenylethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-fluoropyridine
N-(propan-2-yl)-3-(1H-pyrazol-3-yl)benzamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-amine
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
(4aR,8aR)-2-cyclopentanecarbonyl-7-(6-methylpyrimidin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-[2-(morpholin-4-yl)ethyl]urea
N1,N1-dimethyl-N3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-1,3-dicarboxamide
2-amino-4-(2,2-dimethyloxan-4-yl)-6-[4-(morpholin-4-yl)phenyl]pyridine-3-carbonitrile
N-[(3R)-piperidin-3-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]-N-methylpentanamide
9-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)-1,4,9-triazaspiro[5.5]undecan-5-one
5-[4-(2-ethylphenyl)piperazine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
ethyl 2-{[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl](methyl)amino}acetate
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
2-{4-[(5-cyclohexylthiophen-2-yl)methyl]piperazin-1-yl}-N-ethylacetamide
5-ethyl-2-methyl-4-(4-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}piperazin-1-yl)pyrimidine
(2R,6R)-11-methoxy-4-(thiophen-3-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[2-(1H-1,2,4-triazol-1-yl)ethyl]acetamide
N-[cyclopropyl(pyridin-2-yl)methyl]-7-fluoro-N,3-dimethyl-1-benzofuran-2-carboxamide
4-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-N-methylbenzene-1-sulfonamide