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2-{3-[({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}amino)methyl]-2-methyl-1H-indol-1-yl}acetamide
3-{1-[2-(8-methoxy-2H-chromen-3-yl)-1H-imidazol-1-yl]ethyl}-4-propyl-4H-1,2,4-triazole
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-methylpropanamide
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
5-ethyl-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidin-2-amine
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,1-dioxo-1λ6-thiolane-3-carboxamide
(1S,4S)-2-(2H-1,3-benzodioxol-5-yl)-5-[2-(2-chlorophenoxy)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(furan-2-ylmethyl)-1-methyl-3-(2-methylpropyl)-N-(thiophen-2-ylmethyl)-1H-pyrazole-5-carboxamide
7-(pyridin-3-ylmethyl)-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-[(4-fluorophenyl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-(prop-2-en-1-yl)acetamide
(4aR,8aS)-1-[(4-fluorophenyl)methyl]-6-[(2-hydroxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
8-(butane-1-sulfonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[1-(naphthalene-1-carbonyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
4-ethyl-N,N-dimethyl-6-(4-{[1-(pyridin-4-yl)propyl]amino}piperidin-1-yl)pyrimidin-2-amine
(2E)-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-(4-methoxyphenyl)prop-2-enamide
N-tert-butyl-2-[5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]benzene-1-sulfonamide
9-ethyl-1-methyl-4-(3-phenylpropanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-({[2-(2-chlorophenyl)ethyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
N-{2-methoxy-5-[2-(1H-1,2,4-triazol-1-yl)propanamido]phenyl}pentanamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methoxybutanamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-cyclopropyl-1-(2-phenoxybenzoyl)piperazine-2-carboxamide
1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-(3-methylthiophen-2-yl)-1H-1,2,3-triazole
4-[(2S)-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidine-2-carbonyl]morpholine
1-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
N-methyl-4-(4-methylpiperazin-1-yl)-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
2-(4-{[cyclopropyl(1,3-thiazol-5-ylmethyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
2-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-(8-methoxyquinolin-5-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
1-{2-[(5-fluoroquinazolin-4-yl)amino]ethyl}piperidine-3-carboxamide
6-[(diethylamino)methyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-benzyl-5-{[(2-chlorophenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[(2-cyclohexylpyrimidin-5-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
3-{1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]azetidin-3-yl}pyridine
8-[5-(methoxymethyl)furan-2-carbonyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[(3S)-1-benzylpyrrolidin-3-yl]-1-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(dimethylamino)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)quinoxaline-6-carboxamide
3-(2,4-dimethoxyphenyl)-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]-1,2,4-oxadiazole
2-(3-methoxypropyl)-9-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(3-chloro-4-methoxyphenyl)-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
3-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}piperidin-3-yl)benzoic acid
4-{2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-N-[2-(dimethylamino)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine