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3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]propanamide
2-(pyridin-4-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]pyrimidine-5-carboxamide
3-benzyl-1-(3-methoxypropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[(3aS,6aS)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}pyridin-2-amine
4-(3,4-dimethoxyphenyl)-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-ethyl-9-(2-hydroxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(5-{[methyl(oxan-4-yl)amino]methyl}pyrimidin-2-yl)benzenesulfonamide
3-[(dimethylamino)methyl]-N-[2-(4-phenylpiperidin-1-yl)ethyl]benzamide
1-benzoyl-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine
(2S,4R)-4-(dimethylamino)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxylic acid
(1R,5R)-6-[4-(furan-2-yl)benzoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl)[(4-phenoxyphenyl)methyl]amine
2-(3-phenylpropyl)-4-(pyridine-3-sulfonyl)morpholine
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-(propan-2-yl)-2-(1H-pyrazol-1-yl)benzamide
(1s,4s)-4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]cyclohexan-1-ol
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
6-(4-chloro-2-methoxybenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-hexyl-8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-ethoxy-5-{2-[(3-hydroxy-2,2-dimethylpropyl)amino]pyrimidin-4-yl}benzoic acid
3-ethyl-8-(2-methoxypyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-6-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
4-[(2R)-2-amino-3-methoxypropanoyl]-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
3,5-dimethoxy-2-[(4-methoxypiperidin-1-yl)methyl]benzoic acid
1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-(thiomorpholin-4-yl)propan-1-one
6-(2-chlorophenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[(3aS,6aS)-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-octahydropyrrolo[3,4-b]pyrrole-1-carbonyl]morpholine
4-fluoro-2-methyl-N-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzene-1-sulfonamide
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
9-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1H-1,3-benzodiazol-1-yl)-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-[(4-cyclopentylpyrimidin-2-yl)(methyl)amino]-2-methylbutan-2-ol
(2-methoxyethyl)({[2-(2-methylphenyl)pyrimidin-5-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
N-(3,4-difluorophenyl)-1-(furan-3-carbonyl)piperidin-3-amine
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
3-{[6-(dimethylamino)pyrimidin-4-yl]amino}-1-methylpyrrolidin-2-one
3-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
5-[(2,3-dihydro-1H-inden-2-yl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-fluoro-2-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperazin-1-yl}-4-(pyrrolidin-1-yl)pyrimidine
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
2-(5-acetylthiophen-3-yl)-N-[cyclopropyl(4-methylpyridin-2-yl)methyl]acetamide
2-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-N-(propan-2-yl)acetamide
4-hydroxy-N-[2-(1H-indol-1-yl)ethyl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
2-methoxy-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
[2-(2-fluorophenyl)ethyl]({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
2-[4-({[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}methyl)phenyl]ethan-1-amine
2-(2-chlorophenyl)-1-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
N1,N1-dimethyl-N3-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidine-1,3-dicarboxamide
[(1-methyl-1H-imidazol-2-yl)methyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine